VX-745 KINOMEscan - Dataset (ID:20178)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
VX-745 | MK14 | 2.8 | nM |
VX-745 | MK11 | 74.0 | nM |
VX-745 | DDR1 | 1100.0 | nM |
VX-745 | FGR | 1300.0 | nM |
VX-745 | YES | 1600.0 | nM |
VX-745 | LYN | 1700.0 | nM |
VX-745 | ABL2 | 1900.0 | nM |
VX-745 | FYN | 2100.0 | nM |
VX-745 | CSF1R | 2600.0 | nM |
VX-745 | BLK | 3100.0 | nM |
VX-745 | LCK | 4600.0 | nM |
VX-745 | EPHA1 | 4700.0 | nM |
VX-745 | SRC | 5500.0 | nM |
VX-745 | EPHB1 | 6200.0 | nM |
VX-745 | PGFRB | 8400.0 | nM |
VX-745 | PGFRA | 8800.0 | nM |
VX-745 | ABL1-nonphosphorylated | nM | |
VX-745 | ABL1(Y253F)-phosphorylated | nM | |
VX-745 | ABL1(H396P)-nonphosphorylated | nM | |
VX-745 | ABL1(T315I)-phosphorylated | nM | |
VX-745 | ADCK4 | nM | |
VX-745 | ABL1(T315I)-nonphosphorylated | nM | |
VX-745 | ABL1(F317L)-phosphorylated | nM | |
VX-745 | ABL1(F317I)-nonphosphorylated | nM | |
VX-745 | ADCK3 | nM |