SB-203580 KINOMEscan - Dataset (ID:20177)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
SB 203580 | YANK1 | 1300.0 | nM |
SB 203580 | EGFR(L858R,T790M) | 1300.0 | nM |
SB 203580 | EGFR(G719S) | 1300.0 | nM |
SB 203580 | MP2K5 | 1400.0 | nM |
SB 203580 | MK12 | 1500.0 | nM |
SB 203580 | EGFR(L747-T751del,Sins) | 1500.0 | nM |
SB 203580 | EGFR(L747-S752del, P753S) | 1600.0 | nM |
SB 203580 | GSK3B | 1700.0 | nM |
SB 203580 | EGFR(L747-E749del, A750P) | 1700.0 | nM |
SB 203580 | EGFR | 1700.0 | nM |
SB 203580 | CSNK1A1L | 1700.0 | nM |
SB 203580 | FRK | 1800.0 | nM |
SB 203580 | TGFBR2 | 1800.0 | nM |
SB 203580 | EGFR(L858R) | 1900.0 | nM |
SB 203580 | EGFR(S752-I759del) | 2000.0 | nM |
SB 203580 | TYK2(JH2domain-pseudokinase) | 2000.0 | nM |
SB 203580 | YANK2 | 2100.0 | nM |
SB 203580 | TTK | 2500.0 | nM |
SB 203580 | EGFR(T790M) | 2500.0 | nM |
SB 203580 | ABL1(H396P)-nonphosphorylated | 2600.0 | nM |
SB 203580 | PIP5K1C | 2600.0 | nM |
SB 203580 | MRCKB | 2700.0 | nM |
SB 203580 | LCK | 2800.0 | nM |
SB 203580 | ACVR1B | 3000.0 | nM |
SB 203580 | ADCK4 | 3100.0 | nM |