SB-203580 KINOMEscan - Dataset (ID:20177)

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Small Molecule Protein Kd Conc unit
SB 203580 YANK1 1300.0
nM
SB 203580 EGFR(L858R,T790M) 1300.0
nM
SB 203580 EGFR(G719S) 1300.0
nM
SB 203580 MP2K5 1400.0
nM
SB 203580 MK12 1500.0
nM
SB 203580 EGFR(L747-T751del,Sins) 1500.0
nM
SB 203580 EGFR(L747-S752del, P753S) 1600.0
nM
SB 203580 GSK3B 1700.0
nM
SB 203580 EGFR(L747-E749del, A750P) 1700.0
nM
SB 203580 EGFR 1700.0
nM
SB 203580 CSNK1A1L 1700.0
nM
SB 203580 FRK 1800.0
nM
SB 203580 TGFBR2 1800.0
nM
SB 203580 EGFR(L858R) 1900.0
nM
SB 203580 EGFR(S752-I759del) 2000.0
nM
SB 203580 TYK2(JH2domain-pseudokinase) 2000.0
nM
SB 203580 YANK2 2100.0
nM
SB 203580 TTK 2500.0
nM
SB 203580 EGFR(T790M) 2500.0
nM
SB 203580 ABL1(H396P)-nonphosphorylated 2600.0
nM
SB 203580 PIP5K1C 2600.0
nM
SB 203580 MRCKB 2700.0
nM
SB 203580 LCK 2800.0
nM
SB 203580 ACVR1B 3000.0
nM
SB 203580 ADCK4 3100.0
nM