SB-203580 KINOMEscan - Dataset (ID:20177)

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Small Molecule Protein Kd Conc unit
SB 203580 EGFR(T790M) 2500.0
nM
SB 203580 YANK2 2100.0
nM
SB 203580 TYK2(JH2domain-pseudokinase) 2000.0
nM
SB 203580 EGFR(S752-I759del) 2000.0
nM
SB 203580 EGFR(L858R) 1900.0
nM
SB 203580 FRK 1800.0
nM
SB 203580 TGFBR2 1800.0
nM
SB 203580 EGFR 1700.0
nM
SB 203580 CSNK1A1L 1700.0
nM
SB 203580 EGFR(L747-E749del, A750P) 1700.0
nM
SB 203580 GSK3B 1700.0
nM
SB 203580 EGFR(L747-S752del, P753S) 1600.0
nM
SB 203580 MK12 1500.0
nM
SB 203580 EGFR(L747-T751del,Sins) 1500.0
nM
SB 203580 MP2K5 1400.0
nM
SB 203580 YANK1 1300.0
nM
SB 203580 STK36 1300.0
nM
SB 203580 EGFR(L858R,T790M) 1300.0
nM
SB 203580 EGFR(G719S) 1300.0
nM
SB 203580 EPHA6 1200.0
nM
SB 203580 JNK1 1100.0
nM
SB 203580 DDR1 1000.0
nM
SB 203580 RAF1 980.0
nM
SB 203580 PFCDPK1(P.falciparum) 850.0
nM
SB 203580 TNIK 820.0
nM