SB-203580 KINOMEscan - Dataset (ID:20177)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
SB 203580 | EGFR(T790M) | 2500.0 | nM |
SB 203580 | YANK2 | 2100.0 | nM |
SB 203580 | TYK2(JH2domain-pseudokinase) | 2000.0 | nM |
SB 203580 | EGFR(S752-I759del) | 2000.0 | nM |
SB 203580 | EGFR(L858R) | 1900.0 | nM |
SB 203580 | FRK | 1800.0 | nM |
SB 203580 | TGFBR2 | 1800.0 | nM |
SB 203580 | EGFR | 1700.0 | nM |
SB 203580 | CSNK1A1L | 1700.0 | nM |
SB 203580 | EGFR(L747-E749del, A750P) | 1700.0 | nM |
SB 203580 | GSK3B | 1700.0 | nM |
SB 203580 | EGFR(L747-S752del, P753S) | 1600.0 | nM |
SB 203580 | MK12 | 1500.0 | nM |
SB 203580 | EGFR(L747-T751del,Sins) | 1500.0 | nM |
SB 203580 | MP2K5 | 1400.0 | nM |
SB 203580 | YANK1 | 1300.0 | nM |
SB 203580 | STK36 | 1300.0 | nM |
SB 203580 | EGFR(L858R,T790M) | 1300.0 | nM |
SB 203580 | EGFR(G719S) | 1300.0 | nM |
SB 203580 | EPHA6 | 1200.0 | nM |
SB 203580 | JNK1 | 1100.0 | nM |
SB 203580 | DDR1 | 1000.0 | nM |
SB 203580 | RAF1 | 980.0 | nM |
SB 203580 | PFCDPK1(P.falciparum) | 850.0 | nM |
SB 203580 | TNIK | 820.0 | nM |