GSK-1363089 KINOMEscan - Dataset - HMS LINCS Database

GSK-1363089 KINOMEscan - Dataset (ID:20176)

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Small molecules	Proteins

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Small Molecule	Protein	Kd	Conc unit
Foretinib	MKNK1	72.0	nM
Foretinib	MKNK2	3.7	nM
Foretinib	MLCK	3000.0	nM
Foretinib	MLK1	1000.0	nM
Foretinib	MLK2	530.0	nM
Foretinib	MLK3	340.0	nM
Foretinib	MRCKA	660.0	nM
Foretinib	MRCKB	330.0	nM
Foretinib	MST1	1100.0	nM
Foretinib	MST1R	3.0	nM
Foretinib	MST2		nM
Foretinib	MST3		nM
Foretinib	MST4		nM
Foretinib	MTOR		nM
Foretinib	MUSK	13.0	nM
Foretinib	MYLK		nM
Foretinib	MYLK2	2300.0	nM
Foretinib	MYLK4		nM
Foretinib	MYO3A	2800.0	nM
Foretinib	MYO3B	690.0	nM
Foretinib	NDR1		nM
Foretinib	NDR2		nM
Foretinib	NEK1		nM
Foretinib	NEK11		nM
Foretinib	NEK2		nM
Foretinib	NEK3		nM
Foretinib	NEK4		nM
Foretinib	NEK5		nM
Foretinib	NEK6		nM
Foretinib	NEK7		nM
Foretinib	NEK9	470.0	nM
Foretinib	NIM1		nM
Foretinib	NLK	170.0	nM
Foretinib	OSR1		nM
Foretinib	MK14	320.0	nM
Foretinib	MK11	760.0	nM
Foretinib	MK13	54.0	nM
Foretinib	MK12	390.0	nM
Foretinib	PAK1		nM
Foretinib	PAK2		nM
Foretinib	PAK3	4100.0	nM
Foretinib	PAK4		nM
Foretinib	PAK6		nM
Foretinib	PAK7		nM
Foretinib	CDK16	890.0	nM
Foretinib	PCTK2	170.0	nM
Foretinib	PCTK3	250.0	nM
Foretinib	PGFRA	4.5	nM
Foretinib	PGFRB	1.0	nM
Foretinib	PDPK1		nM
Foretinib	PFCDPK1(P.falciparum)	230.0	nM
Foretinib	PFPK5(P.falciparum)		nM
Foretinib	CDK15	32.0	nM
Foretinib	CDK14	31.0	nM
Foretinib	PHKG1		nM
Foretinib	PHKG2		nM
Foretinib	PIK3C2B		nM
Foretinib	PIK3C2G		nM
Foretinib	PIK3CA		nM
Foretinib	PIK3CA(C420R)		nM
Foretinib	PIK3CA(E542K)		nM
Foretinib	PIK3CA(E545A)		nM
Foretinib	PIK3CA(E545K)		nM
Foretinib	PIK3CA(H1047L)		nM
Foretinib	PIK3CA(H1047Y)		nM
Foretinib	PIK3CA(I800L)		nM
Foretinib	PIK3CA(M1043I)		nM
Foretinib	PIK3CA(Q546K)		nM
Foretinib	PIK3CB		nM
Foretinib	PIK3CD		nM
Foretinib	PIK3CG		nM
Foretinib	PIK4CB		nM
Foretinib	PIM1		nM
Foretinib	PIM2		nM
Foretinib	PIM3		nM
Foretinib	PIP5K1A		nM
Foretinib	PIP5K1C		nM
Foretinib	PIP5K2B		nM
Foretinib	PI42C	28.0	nM
Foretinib	PKAC-alpha		nM
Foretinib	PKAC-beta		nM
Foretinib	PKMYT1		nM
Foretinib	PKN1		nM
Foretinib	PKN2		nM
Foretinib	PKNB(M.tuberculosis)		nM
Foretinib	PLK1		nM
Foretinib	PLK2		nM
Foretinib	PLK3		nM
Foretinib	PLK4	3.5	nM
Foretinib	KPCD		nM
Foretinib	KPCE		nM
Foretinib	KPCL		nM
Foretinib	KPCI		nM
Foretinib	KPCT		nM
Foretinib	KPCD1		nM
Foretinib	KPCD2		nM
Foretinib	KPCD3	7500.0	nM
Foretinib	KGP1		nM
Foretinib	KGP2		nM
Foretinib	PRKR		nM
Foretinib	PRKX		nM
Foretinib	PRP4		nM
Foretinib	FAK2	14.0	nM
Foretinib	SIK3		nM
Foretinib	RAF1	4400.0	nM
Foretinib	RET	0.7	nM
Foretinib	RET(M918T)	0.7	nM
Foretinib	RET(V804L)	1.6	nM
Foretinib	RET(V804M)	2.8	nM
Foretinib	RIOK1		nM
Foretinib	RIOK2		nM
Foretinib	RIOK3		nM
Foretinib	RIPK1	850.0	nM
Foretinib	RIPK2	21.0	nM
Foretinib	RIPK4	900.0	nM
Foretinib	RIPK5	510.0	nM
Foretinib	ROCK1		nM
Foretinib	ROCK2	1800.0	nM
Foretinib	ROS1	14.0	nM
Foretinib	RPS6KA4(Kin.Dom.1-N-terminal)		nM
Foretinib	RPS6KA4(Kin.Dom.2-C-terminal)		nM
Foretinib	RPS6KA5(Kin.Dom.1-N-terminal)		nM
Foretinib	RPS6KA5(Kin.Dom.2-C-terminal)		nM
Foretinib	RSK1(Kin.Dom.1-N-terminal)		nM
Foretinib	RSK1(Kin.Dom.2-C-terminal)		nM
Foretinib	RSK2(Kin.Dom.1-N-terminal)		nM
Foretinib	RSK3(Kin.Dom.1-N-terminal)	5100.0	nM
Foretinib	RSK3(Kin.Dom.2-C-terminal)		nM
Foretinib	RSK4(Kin.Dom.1-N-terminal)		nM
Foretinib	RSK4(Kin.Dom.2-C-terminal)		nM
Foretinib	S6K1	1200.0	nM
Foretinib	SBK1		nM
Foretinib	SgK110		nM
Foretinib	SGK3		nM
Foretinib	SIK1	160.0	nM
Foretinib	SIK2	640.0	nM
Foretinib	SLK	3.0	nM
Foretinib	SNARK		nM
Foretinib	SNRK		nM
Foretinib	SRC	20.0	nM
Foretinib	SRMS	18.0	nM
Foretinib	SRPK1		nM
Foretinib	SRPK2		nM
Foretinib	SRPK3		nM
Foretinib	STK16		nM
Foretinib	STK33	98.0	nM
Foretinib	STK35	230.0	nM
Foretinib	STK36	180.0	nM
Foretinib	STK39		nM
Foretinib	SYK	280.0	nM
Foretinib	TAK1	540.0	nM
Foretinib	TAOK1	3700.0	nM
Foretinib	TAOK2	6900.0	nM
Foretinib	TAOK3		nM
Foretinib	TBK1	800.0	nM
Foretinib	TEC	310.0	nM
Foretinib	TESK1	260.0	nM
Foretinib	TGFBR1		nM
Foretinib	TGFBR2		nM
Foretinib	TIE1	0.8	nM
Foretinib	TIE2	3.1	nM
Foretinib	TLK1		nM
Foretinib	TLK2		nM
Foretinib	TNIK	210.0	nM
Foretinib	TNK1	21.0	nM
Foretinib	TNK2	200.0	nM
Foretinib	TNNI3K	130.0	nM
Foretinib	TRKA	4.8	nM
Foretinib	TRKB	4.1	nM
Foretinib	TRKC	3.4	nM
Foretinib	TRPM6		nM
Foretinib	TSSK1		nM
Foretinib	TTK	430.0	nM
Foretinib	TXK	530.0	nM
Foretinib	TYK2(JH1domain-catalytic)	5000.0	nM
Foretinib	TYK2(JH2domain-pseudokinase)		nM
Foretinib	TYRO3	2.0	nM
Foretinib	ULK1		nM
Foretinib	ULK2		nM
Foretinib	ULK3	450.0	nM
Foretinib	VGFR2	12.0	nM
Foretinib	VRK2		nM
Foretinib	WEE1		nM
Foretinib	WEE2		nM
Foretinib	YANK1		nM
Foretinib	YANK2		nM
Foretinib	YANK3		nM
Foretinib	YES	48.0	nM
Foretinib	YSK1	5700.0	nM
Foretinib	YSK4	5.5	nM
Foretinib	MLTK	45.0	nM
Foretinib	ZAP70		nM

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HMS LINCS Project

GSK-1363089 KINOMEscan - Dataset (ID:20176)