GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Foretinib | IKKB | nM | |
Foretinib | IKKE | 1400.0 | nM |
Foretinib | INSR | 210.0 | nM |
Foretinib | INSRR | 53.0 | nM |
Foretinib | IRAK1 | nM | |
Foretinib | IRAK3 | 370.0 | nM |
Foretinib | IRAK4 | nM | |
Foretinib | ITK | 69.0 | nM |
Foretinib | JAK1(JH1domain-catalytic) | nM | |
Foretinib | JAK1(JH2domain-pseudokinase) | nM | |
Foretinib | JAK2(JH1domain-catalytic) | 1500.0 | nM |
Foretinib | JAK3(JH1domain-catalytic) | nM | |
Foretinib | JNK1 | 5700.0 | nM |
Foretinib | JNK3 | 3900.0 | nM |
Foretinib | KC1G1 | nM | |
Foretinib | KC1G2 | nM | |
Foretinib | KCC2D | nM | |
Foretinib | KCC4 | nM | |
Foretinib | KGP1 | nM | |
Foretinib | KGP2 | nM | |
Foretinib | KIT | 2.5 | nM |
Foretinib | KIT(A829P) | 3.2 | nM |
Foretinib | KIT(D816H) | 36.0 | nM |
Foretinib | KIT(D816V) | 9.6 | nM |
Foretinib | KIT(L576P) | 2.7 | nM |