GSK-1363089 KINOMEscan - Dataset (ID:20176)

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Small Molecule Protein Kd Conc unit
Foretinib CAMK2B
nM
Foretinib CAMK2G
nM
Foretinib CAMKK2 4400.0
nM
Foretinib CASK
nM
Foretinib CDC2L1 640.0
nM
Foretinib CDC2L2 480.0
nM
Foretinib CDC2L5 210.0
nM
Foretinib CDK11 87.0
nM
Foretinib CDK14 31.0
nM
Foretinib CDK15 32.0
nM
Foretinib CDK16 890.0
nM
Foretinib CDK2
nM
Foretinib CDK3
nM
Foretinib CDK4-cyclinD1
nM
Foretinib CDK4-cyclinD3
nM
Foretinib CDK5
nM
Foretinib CDK7 3.7
nM
Foretinib CDK8 130.0
nM
Foretinib CDK9 1600.0
nM
Foretinib CDKL1
nM
Foretinib CDKL2 240.0
nM
Foretinib CDKL3 4400.0
nM
Foretinib CDKL5 2700.0
nM
Foretinib CHEK1
nM
Foretinib CHK2 57.0
nM