GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Foretinib | MINK | 2600.0 | nM |
Foretinib | BRAF(V600E) | 2300.0 | nM |
Foretinib | MYLK2 | 2300.0 | nM |
Foretinib | DYRK2 | 2000.0 | nM |
Foretinib | MAP4K2 | 2000.0 | nM |
Foretinib | M3K2 | 1900.0 | nM |
Foretinib | MAP3K4 | 1900.0 | nM |
Foretinib | MAK | 1800.0 | nM |
Foretinib | ROCK2 | 1800.0 | nM |
Foretinib | EGFR(L858R,T790M) | 1800.0 | nM |
Foretinib | LIMK2 | 1700.0 | nM |
Foretinib | CDK9 | 1600.0 | nM |
Foretinib | FGFR3(G697C) | 1600.0 | nM |
Foretinib | ANKK1 | 1500.0 | nM |
Foretinib | JAK2(JH1domain-catalytic) | 1500.0 | nM |
Foretinib | ERBB3 | 1500.0 | nM |
Foretinib | IKKE | 1400.0 | nM |
Foretinib | AMPK-alpha2 | 1200.0 | nM |
Foretinib | S6K1 | 1200.0 | nM |
Foretinib | EGFR(S752-I759del) | 1100.0 | nM |
Foretinib | MST1 | 1100.0 | nM |
Foretinib | MLK1 | 1000.0 | nM |
Foretinib | EIF2AK1 | 980.0 | nM |
Foretinib | FGFR3 | 910.0 | nM |
Foretinib | RIPK4 | 900.0 | nM |