GSK-1363089 KINOMEscan - Dataset (ID:20176)

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Small Molecule Protein Kd Conc unit
Foretinib MINK 2600.0
nM
Foretinib BRAF(V600E) 2300.0
nM
Foretinib MYLK2 2300.0
nM
Foretinib DYRK2 2000.0
nM
Foretinib MAP4K2 2000.0
nM
Foretinib M3K2 1900.0
nM
Foretinib MAP3K4 1900.0
nM
Foretinib MAK 1800.0
nM
Foretinib ROCK2 1800.0
nM
Foretinib EGFR(L858R,T790M) 1800.0
nM
Foretinib LIMK2 1700.0
nM
Foretinib CDK9 1600.0
nM
Foretinib FGFR3(G697C) 1600.0
nM
Foretinib ANKK1 1500.0
nM
Foretinib JAK2(JH1domain-catalytic) 1500.0
nM
Foretinib ERBB3 1500.0
nM
Foretinib IKKE 1400.0
nM
Foretinib AMPK-alpha2 1200.0
nM
Foretinib S6K1 1200.0
nM
Foretinib EGFR(S752-I759del) 1100.0
nM
Foretinib MST1 1100.0
nM
Foretinib MLK1 1000.0
nM
Foretinib EIF2AK1 980.0
nM
Foretinib FGFR3 910.0
nM
Foretinib RIPK4 900.0
nM