GSK-1363089 KINOMEscan - Dataset (ID:20176)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Foretinib | DCAMKL2 | nM | |
| Foretinib | DCAMKL3 | nM | |
| Foretinib | DDR1 | 0.2 | nM |
| Foretinib | DDR2 | 3.6 | nM |
| Foretinib | M3K12 | 22.0 | nM |
| Foretinib | DMPK | nM | |
| Foretinib | DMPK2 | 180.0 | nM |
| Foretinib | DRAK1 | nM | |
| Foretinib | DRAK2 | nM | |
| Foretinib | DYRK1A | nM | |
| Foretinib | DYRK1B | nM | |
| Foretinib | DYRK2 | 2000.0 | nM |
| Foretinib | EGFR | 440.0 | nM |
| Foretinib | EGFR(E746-A750del) | 310.0 | nM |
| Foretinib | EGFR(G719C) | 120.0 | nM |
| Foretinib | EGFR(G719S) | 370.0 | nM |
| Foretinib | EGFR(L747-E749del, A750P) | 160.0 | nM |
| Foretinib | EGFR(L747-S752del, P753S) | 210.0 | nM |
| Foretinib | EGFR(L747-T751del,Sins) | 160.0 | nM |
| Foretinib | EGFR(L858R) | 190.0 | nM |
| Foretinib | EGFR(L858R,T790M) | 1800.0 | nM |
| Foretinib | EGFR(L861Q) | 86.0 | nM |
| Foretinib | EGFR(S752-I759del) | 1100.0 | nM |
| Foretinib | EGFR(T790M) | 470.0 | nM |
| Foretinib | EIF2AK1 | 980.0 | nM |