BIBF-1120 KINOMEscan - Dataset (ID:20175)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Nintedanib | M3K2 | 9.4 | nM |
Nintedanib | RET(V804M) | 9.6 | nM |
Nintedanib | RET(V804L) | 9.8 | nM |
Nintedanib | ABL1(T315I)-phosphorylated | 10.0 | nM |
Nintedanib | MP2K1 | 10.0 | nM |
Nintedanib | DDR1 | 12.0 | nM |
Nintedanib | SRPK3 | 12.0 | nM |
Nintedanib | AXL | 12.0 | nM |
Nintedanib | JAK2(JH1domain-catalytic) | 14.0 | nM |
Nintedanib | KGP1 | 14.0 | nM |
Nintedanib | PGFRB | 15.0 | nM |
Nintedanib | PGFRA | 16.0 | nM |
Nintedanib | FLT3(R834Q) | 17.0 | nM |
Nintedanib | PIP5K2B | 17.0 | nM |
Nintedanib | GRK4 | 17.0 | nM |
Nintedanib | LKB1 | 18.0 | nM |
Nintedanib | STK16 | 18.0 | nM |
Nintedanib | CLK4 | 18.0 | nM |
Nintedanib | TRKB | 19.0 | nM |
Nintedanib | SNARK | 21.0 | nM |
Nintedanib | INSRR | 21.0 | nM |
Nintedanib | CDK16 | 21.0 | nM |
Nintedanib | TTK | 22.0 | nM |
Nintedanib | RIOK1 | 23.0 | nM |
Nintedanib | INSR | 24.0 | nM |