BIBF-1120 KINOMEscan - Dataset (ID:20175)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Nintedanib | KIT(L576P) | 2.7 | nM |
Nintedanib | FLT3(N841I) | 2.6 | nM |
Nintedanib | BIKE | 2.2 | nM |
Nintedanib | MP2K5 | 1.8 | nM |
Nintedanib | FLT3(D835H) | 0.7 | nM |
Nintedanib | FLT3(ITD) | 0.7 | nM |
Nintedanib | FLT3(D835Y) | 0.4 | nM |
Nintedanib | KC1G2 | nM | |
Nintedanib | KC1G1 | nM | |
Nintedanib | CSNK1A1L | nM | |
Nintedanib | CSNK1A1 | nM | |
Nintedanib | CSK | nM | |
Nintedanib | PFPK5(P.falciparum) | nM | |
Nintedanib | CDK15 | nM | |
Nintedanib | CLK3 | nM | |
Nintedanib | PIK3C2B | nM | |
Nintedanib | PIK3C2G | nM | |
Nintedanib | PIK3CA | nM | |
Nintedanib | PIK3CA(C420R) | nM | |
Nintedanib | PIK3CA(E542K) | nM | |
Nintedanib | PIK3CA(E545A) | nM | |
Nintedanib | PIK3CA(E545K) | nM | |
Nintedanib | PIK3CA(H1047L) | nM | |
Nintedanib | PIK3CA(H1047Y) | nM | |
Nintedanib | PIK3CA(I800L) | nM |