BIBF-1120 KINOMEscan - Dataset (ID:20175)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Nintedanib | IKKB | nM | |
Nintedanib | IKKE | 170.0 | nM |
Nintedanib | INSR | 24.0 | nM |
Nintedanib | INSRR | 21.0 | nM |
Nintedanib | IRAK1 | 120.0 | nM |
Nintedanib | IRAK3 | 5300.0 | nM |
Nintedanib | IRAK4 | 810.0 | nM |
Nintedanib | ITK | 210.0 | nM |
Nintedanib | JAK1(JH1domain-catalytic) | 2500.0 | nM |
Nintedanib | JAK1(JH2domain-pseudokinase) | 4.8 | nM |
Nintedanib | JAK2(JH1domain-catalytic) | 14.0 | nM |
Nintedanib | JAK3(JH1domain-catalytic) | 8.2 | nM |
Nintedanib | JNK1 | 630.0 | nM |
Nintedanib | JNK3 | 270.0 | nM |
Nintedanib | KC1G1 | nM | |
Nintedanib | KC1G2 | nM | |
Nintedanib | KCC2D | nM | |
Nintedanib | KCC4 | 3700.0 | nM |
Nintedanib | KGP1 | 14.0 | nM |
Nintedanib | KGP2 | nM | |
Nintedanib | KIT | 5.7 | nM |
Nintedanib | KIT(A829P) | 87.0 | nM |
Nintedanib | KIT(D816H) | 310.0 | nM |
Nintedanib | KIT(D816V) | 47.0 | nM |
Nintedanib | KIT(L576P) | 2.7 | nM |