BIBF-1120 KINOMEscan - Dataset (ID:20175)

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Small Molecule Protein Kd Conc unit
Nintedanib IKKB
nM
Nintedanib IKKE 170.0
nM
Nintedanib INSR 24.0
nM
Nintedanib INSRR 21.0
nM
Nintedanib IRAK1 120.0
nM
Nintedanib IRAK3 5300.0
nM
Nintedanib IRAK4 810.0
nM
Nintedanib ITK 210.0
nM
Nintedanib JAK1(JH1domain-catalytic) 2500.0
nM
Nintedanib JAK1(JH2domain-pseudokinase) 4.8
nM
Nintedanib JAK2(JH1domain-catalytic) 14.0
nM
Nintedanib JAK3(JH1domain-catalytic) 8.2
nM
Nintedanib JNK1 630.0
nM
Nintedanib JNK3 270.0
nM
Nintedanib KC1G1
nM
Nintedanib KC1G2
nM
Nintedanib KCC2D
nM
Nintedanib KCC4 3700.0
nM
Nintedanib KGP1 14.0
nM
Nintedanib KGP2
nM
Nintedanib KIT 5.7
nM
Nintedanib KIT(A829P) 87.0
nM
Nintedanib KIT(D816H) 310.0
nM
Nintedanib KIT(D816V) 47.0
nM
Nintedanib KIT(L576P) 2.7
nM