BIBF-1120 KINOMEscan - Dataset (ID:20175)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Nintedanib | KIT | 5.7 | nM |
Nintedanib | KIT(A829P) | 87.0 | nM |
Nintedanib | KIT(D816H) | 310.0 | nM |
Nintedanib | KIT(D816V) | 47.0 | nM |
Nintedanib | KIT(L576P) | 2.7 | nM |
Nintedanib | KIT(V559D) | 6.3 | nM |
Nintedanib | KIT(V559D,T670I) | 2.9 | nM |
Nintedanib | KIT(V559D,V654A) | 29.0 | nM |
Nintedanib | LATS1 | 420.0 | nM |
Nintedanib | LATS2 | 380.0 | nM |
Nintedanib | LCK | 6.2 | nM |
Nintedanib | LIMK1 | nM | |
Nintedanib | LIMK2 | nM | |
Nintedanib | LKB1 | 18.0 | nM |
Nintedanib | LOK | 87.0 | nM |
Nintedanib | LRRK2 | 46.0 | nM |
Nintedanib | LRRK2(G2019S) | 37.0 | nM |
Nintedanib | LTK | 150.0 | nM |
Nintedanib | LYN | 940.0 | nM |
Nintedanib | M3K13 | 140.0 | nM |
Nintedanib | MAK | nM | |
Nintedanib | MAP3K1 | nM | |
Nintedanib | MAP3K15 | 1400.0 | nM |
Nintedanib | M3K2 | 9.4 | nM |
Nintedanib | MAP3K3 | 34.0 | nM |