TKI-258 KINOMEscan - Dataset (ID:20168)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Dovitinib | ZAP70 | nM | |
Dovitinib | YSK4 | 12.0 | nM |
Dovitinib | YSK1 | 1200.0 | nM |
Dovitinib | YES | 580.0 | nM |
Dovitinib | YANK3 | nM | |
Dovitinib | YANK2 | nM | |
Dovitinib | YANK1 | nM | |
Dovitinib | WEE2 | nM | |
Dovitinib | WEE1 | 1200.0 | nM |
Dovitinib | VRK2 | nM | |
Dovitinib | VGFR2 | 68.0 | nM |
Dovitinib | VGFR1 | 69.0 | nM |
Dovitinib | ULK3 | 170.0 | nM |
Dovitinib | ULK2 | 54.0 | nM |
Dovitinib | ULK1 | 55.0 | nM |
Dovitinib | TYRO3 | 9300.0 | nM |
Dovitinib | TYK2(JH2domain-pseudokinase) | 2200.0 | nM |
Dovitinib | TYK2(JH1domain-catalytic) | 150.0 | nM |
Dovitinib | TXK | nM | |
Dovitinib | TTK | nM | |
Dovitinib | TSSK1 | nM | |
Dovitinib | TRPM6 | nM | |
Dovitinib | TRKC | 190.0 | nM |
Dovitinib | TRKB | 720.0 | nM |
Dovitinib | TRKA | 100.0 | nM |