TKI-258 KINOMEscan - Dataset (ID:20168)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Dovitinib | FES | nM | |
| Dovitinib | FGFR1 | 150.0 | nM |
| Dovitinib | FGFR2 | 410.0 | nM |
| Dovitinib | FGFR3 | 230.0 | nM |
| Dovitinib | FGFR3(G697C) | 370.0 | nM |
| Dovitinib | FGFR4 | 4300.0 | nM |
| Dovitinib | FGR | 190.0 | nM |
| Dovitinib | VGFR1 | 69.0 | nM |
| Dovitinib | FLT3 | 0.6 | nM |
| Dovitinib | FLT3(D835H) | 6.1 | nM |
| Dovitinib | FLT3(D835Y) | 5.2 | nM |
| Dovitinib | FLT3(ITD) | 3.6 | nM |
| Dovitinib | FLT3(K663Q) | 1.1 | nM |
| Dovitinib | FLT3(N841I) | 4.8 | nM |
| Dovitinib | FLT3(R834Q) | 7.5 | nM |
| Dovitinib | FLT4 | 580.0 | nM |
| Dovitinib | FRK | 2300.0 | nM |
| Dovitinib | FYN | 440.0 | nM |
| Dovitinib | GAK | 490.0 | nM |
| Dovitinib | GCN2(Kin.Dom.2,S808G) | 250.0 | nM |
| Dovitinib | GRK1 | 2200.0 | nM |
| Dovitinib | GRK4 | 97.0 | nM |
| Dovitinib | GRK7 | 1300.0 | nM |
| Dovitinib | GSK3A | nM | |
| Dovitinib | GSK3B | 350.0 | nM |