TKI-258 KINOMEscan - Dataset (ID:20168)

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Small Molecule Protein Kd Conc unit
Dovitinib AKT3
nM
Dovitinib ALK 3500.0
nM
Dovitinib AMPK-alpha1 520.0
nM
Dovitinib AMPK-alpha2 820.0
nM
Dovitinib ANKK1 79.0
nM
Dovitinib NUAK1 240.0
nM
Dovitinib M3K5
nM
Dovitinib M3K6
nM
Dovitinib AURKA
nM
Dovitinib AURKB 280.0
nM
Dovitinib AURKC 1100.0
nM
Dovitinib AXL 3800.0
nM
Dovitinib BIKE 54.0
nM
Dovitinib BLK 190.0
nM
Dovitinib BMPR1A
nM
Dovitinib BMPR1B
nM
Dovitinib BMPR2 3100.0
nM
Dovitinib BMX
nM
Dovitinib BRAF
nM
Dovitinib BRAF(V600E)
nM
Dovitinib PTK6
nM
Dovitinib BRSK1
nM
Dovitinib BRSK2
nM
Dovitinib BTK
nM
Dovitinib AAK1 170.0
nM