TKI-258 KINOMEscan - Dataset (ID:20168)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Dovitinib | ABL1(Y253F)-phosphorylated | 46.0 | nM |
Dovitinib | RET(M918T) | 47.0 | nM |
Dovitinib | ABL1(M351T)-phosphorylated | 48.0 | nM |
Dovitinib | ULK2 | 54.0 | nM |
Dovitinib | BIKE | 54.0 | nM |
Dovitinib | PGFRA | 54.0 | nM |
Dovitinib | ABL1-phosphorylated | 54.0 | nM |
Dovitinib | ULK1 | 55.0 | nM |
Dovitinib | ABL1(Q252H)-phosphorylated | 58.0 | nM |
Dovitinib | CSF1R | 60.0 | nM |
Dovitinib | ABL1(H396P)-phosphorylated | 60.0 | nM |
Dovitinib | VGFR2 | 68.0 | nM |
Dovitinib | VGFR1 | 69.0 | nM |
Dovitinib | RET | 71.0 | nM |
Dovitinib | M3K2 | 71.0 | nM |
Dovitinib | ABL1(Q252H)-nonphosphorylated | 75.0 | nM |
Dovitinib | ABL1(E255K)-phosphorylated | 75.0 | nM |
Dovitinib | ANKK1 | 79.0 | nM |
Dovitinib | MYLK4 | 80.0 | nM |
Dovitinib | MYLK2 | 92.0 | nM |
Dovitinib | GRK4 | 97.0 | nM |
Dovitinib | ABL1-nonphosphorylated | 100.0 | nM |
Dovitinib | TRKA | 100.0 | nM |
Dovitinib | ABL1(T315I)-nonphosphorylated | 110.0 | nM |
Dovitinib | JAK2(JH1domain-catalytic) | 130.0 | nM |