TKI-258 KINOMEscan - Dataset (ID:20168)

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Small Molecule Protein Kd Conc unit
Dovitinib HIPK1 4200.0
nM
Dovitinib HIPK2 500.0
nM
Dovitinib HIPK3 5100.0
nM
Dovitinib HIPK4
nM
Dovitinib M4K1 44.0
nM
Dovitinib HUNK 410.0
nM
Dovitinib ICK
nM
Dovitinib IGF1R
nM
Dovitinib IKKA 1800.0
nM
Dovitinib IKKB
nM
Dovitinib IKKE 480.0
nM
Dovitinib INSR
nM
Dovitinib INSRR
nM
Dovitinib IRAK1 170.0
nM
Dovitinib IRAK3
nM
Dovitinib IRAK4 130.0
nM
Dovitinib ITK 530.0
nM
Dovitinib JAK1(JH1domain-catalytic)
nM
Dovitinib JAK1(JH2domain-pseudokinase) 380.0
nM
Dovitinib JAK2(JH1domain-catalytic) 130.0
nM
Dovitinib JAK3(JH1domain-catalytic) 410.0
nM
Dovitinib JNK1
nM
Dovitinib MK09
nM
Dovitinib JNK3
nM
Dovitinib AAK1 170.0
nM