TKI-258 KINOMEscan - Dataset (ID:20168)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Dovitinib | KIT | 7.5 | nM |
| Dovitinib | KIT(A829P) | 45.0 | nM |
| Dovitinib | KIT(D816H) | 170.0 | nM |
| Dovitinib | KIT(D816V) | 1400.0 | nM |
| Dovitinib | KIT(L576P) | 1.6 | nM |
| Dovitinib | KIT(V559D) | 7.2 | nM |
| Dovitinib | KIT(V559D,T670I) | 26.0 | nM |
| Dovitinib | KIT(V559D,V654A) | 3.1 | nM |
| Dovitinib | LATS1 | 1700.0 | nM |
| Dovitinib | LATS2 | 530.0 | nM |
| Dovitinib | LCK | 250.0 | nM |
| Dovitinib | LIMK1 | nM | |
| Dovitinib | LIMK2 | nM | |
| Dovitinib | LKB1 | 3700.0 | nM |
| Dovitinib | LOK | 550.0 | nM |
| Dovitinib | LRRK2 | 1500.0 | nM |
| Dovitinib | LRRK2(G2019S) | 880.0 | nM |
| Dovitinib | LTK | nM | |
| Dovitinib | LYN | 750.0 | nM |
| Dovitinib | M3K13 | 170.0 | nM |
| Dovitinib | MAK | nM | |
| Dovitinib | MAP3K1 | nM | |
| Dovitinib | MAP3K15 | nM | |
| Dovitinib | M3K2 | 71.0 | nM |
| Dovitinib | MAP3K3 | nM |