TKI-258 KINOMEscan - Dataset (ID:20168)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Dovitinib | PRKX | nM | |
| Dovitinib | PRP4 | 560.0 | nM |
| Dovitinib | FAK2 | nM | |
| Dovitinib | SIK3 | nM | |
| Dovitinib | RAF1 | nM | |
| Dovitinib | RET | 71.0 | nM |
| Dovitinib | RET(M918T) | 47.0 | nM |
| Dovitinib | RET(V804L) | 27.0 | nM |
| Dovitinib | RET(V804M) | 26.0 | nM |
| Dovitinib | RIOK1 | 420.0 | nM |
| Dovitinib | RIOK2 | 260.0 | nM |
| Dovitinib | RIOK3 | 690.0 | nM |
| Dovitinib | RIPK1 | 320.0 | nM |
| Dovitinib | RIPK2 | nM | |
| Dovitinib | RIPK4 | nM | |
| Dovitinib | RIPK5 | nM | |
| Dovitinib | ROCK1 | 760.0 | nM |
| Dovitinib | ROCK2 | 3100.0 | nM |
| Dovitinib | ROS1 | nM | |
| Dovitinib | RPS6KA4(Kin.Dom.1-N-terminal) | 590.0 | nM |
| Dovitinib | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
| Dovitinib | RPS6KA5(Kin.Dom.1-N-terminal) | 680.0 | nM |
| Dovitinib | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
| Dovitinib | RSK1(Kin.Dom.1-N-terminal) | 450.0 | nM |
| Dovitinib | RSK1(Kin.Dom.2-C-terminal) | nM |