PI-103 KINOMEscan - Dataset (ID:20167)

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Small Molecule Protein Kd Conc unit
PI103 JAK1(JH2domain-pseudokinase) 2000.0
nM
PI103 BRAF(V600E) 2300.0
nM
PI103 DAPK1 2400.0
nM
PI103 FLT3 2500.0
nM
PI103 DAPK2 2700.0
nM
PI103 BRAF 2900.0
nM
PI103 CSNK2A2 2900.0
nM
PI103 HIPK1 3300.0
nM
PI103 PIK4CB 3500.0
nM
PI103 LIMK2 3500.0
nM
PI103 RAF1 3700.0
nM
PI103 CLK1 3900.0
nM
PI103 DYRK2 4100.0
nM
PI103 CSNK2A1 5400.0
nM
PI103 CLK2 5500.0
nM
PI103 DYRK1B 5700.0
nM
PI103 TYK2(JH2domain-pseudokinase) 5900.0
nM
PI103 FLT3(D835H) 5900.0
nM
PI103 CLK3 5900.0
nM
PI103 FLT3(ITD) 7200.0
nM
PI103 CDK7 7200.0
nM
PI103 ANKK1
nM
PI103 AMPK-alpha2
nM
PI103 ABL1-nonphosphorylated
nM
PI103 AMPK-alpha1
nM