PI-103 KINOMEscan - Dataset (ID:20167)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PI103 | JAK1(JH2domain-pseudokinase) | 2000.0 | nM |
PI103 | BRAF(V600E) | 2300.0 | nM |
PI103 | DAPK1 | 2400.0 | nM |
PI103 | FLT3 | 2500.0 | nM |
PI103 | DAPK2 | 2700.0 | nM |
PI103 | BRAF | 2900.0 | nM |
PI103 | CSNK2A2 | 2900.0 | nM |
PI103 | HIPK1 | 3300.0 | nM |
PI103 | PIK4CB | 3500.0 | nM |
PI103 | LIMK2 | 3500.0 | nM |
PI103 | RAF1 | 3700.0 | nM |
PI103 | CLK1 | 3900.0 | nM |
PI103 | DYRK2 | 4100.0 | nM |
PI103 | CSNK2A1 | 5400.0 | nM |
PI103 | CLK2 | 5500.0 | nM |
PI103 | DYRK1B | 5700.0 | nM |
PI103 | TYK2(JH2domain-pseudokinase) | 5900.0 | nM |
PI103 | FLT3(D835H) | 5900.0 | nM |
PI103 | CLK3 | 5900.0 | nM |
PI103 | FLT3(ITD) | 7200.0 | nM |
PI103 | CDK7 | 7200.0 | nM |
PI103 | ANKK1 | nM | |
PI103 | AMPK-alpha2 | nM | |
PI103 | ABL1-nonphosphorylated | nM | |
PI103 | AMPK-alpha1 | nM |