PI-103 KINOMEscan - Dataset (ID:20167)

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Small Molecule Protein Kd Conc unit
PI103 DAPK3 840.0
nM
PI103 RIOK2 770.0
nM
PI103 PI42C 620.0
nM
PI103 HIPK3 310.0
nM
PI103 HIPK2 290.0
nM
PI103 PIK3C2G 41.0
nM
PI103 PIK3CD 17.0
nM
PI103 PIK3CG 16.0
nM
PI103 MTOR 12.0
nM
PI103 PIK3C2B 10.0
nM
PI103 PIK3CA(H1047Y) 3.4
nM
PI103 PIK3CA(H1047L) 3.2
nM
PI103 PIK3CA(M1043I) 3.0
nM
PI103 PIK3CA(I800L) 2.9
nM
PI103 PIK3CB 1.7
nM
PI103 PIK3CA(Q546K) 1.5
nM
PI103 PIK3CA(E545K) 1.5
nM
PI103 PIK3CA 1.5
nM
PI103 PIK3CA(E545A) 1.5
nM
PI103 PIK3CA(E542K) 1.4
nM
PI103 PIK3CA(C420R) 1.3
nM
PI103 ANKK1
nM
PI103 AMPK-alpha2
nM
PI103 ABL1-nonphosphorylated
nM
PI103 AMPK-alpha1
nM