PI-103 KINOMEscan - Dataset (ID:20167)

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Small Molecule Protein Kd Conc unit
PI103 PFCDPK1(P.falciparum)
nM
PI103 PFPK5(P.falciparum)
nM
PI103 CDK15
nM
PI103 CDK14
nM
PI103 PHKG1
nM
PI103 PHKG2
nM
PI103 PIK3C2B 10.0
nM
PI103 PIK3C2G 41.0
nM
PI103 PIK3CA 1.5
nM
PI103 PIK3CA(C420R) 1.3
nM
PI103 PIK3CA(E542K) 1.4
nM
PI103 PIK3CA(E545A) 1.5
nM
PI103 PIK3CA(E545K) 1.5
nM
PI103 PIK3CA(H1047L) 3.2
nM
PI103 PIK3CA(H1047Y) 3.4
nM
PI103 PIK3CA(I800L) 2.9
nM
PI103 PIK3CA(M1043I) 3.0
nM
PI103 PIK3CA(Q546K) 1.5
nM
PI103 PIK3CB 1.7
nM
PI103 PIK3CD 17.0
nM
PI103 PIK3CG 16.0
nM
PI103 PIK4CB 3500.0
nM
PI103 PIM1
nM
PI103 PIM2
nM
PI103 PIM3
nM