PHA-665752 KINOMEscan - Dataset (ID:20166)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PHA-665752 | MET | 0.3 | nM |
PHA-665752 | MET(M1250T) | 0.6 | nM |
PHA-665752 | MET(Y1235D) | 0.8 | nM |
PHA-665752 | SRPK1 | 41.0 | nM |
PHA-665752 | TAOK3 | 43.0 | nM |
PHA-665752 | BIKE | 47.0 | nM |
PHA-665752 | FLT3(ITD) | 58.0 | nM |
PHA-665752 | GRK7 | 61.0 | nM |
PHA-665752 | HIPK3 | 63.0 | nM |
PHA-665752 | KKCC1 | 64.0 | nM |
PHA-665752 | DDR1 | 70.0 | nM |
PHA-665752 | CAMKK2 | 73.0 | nM |
PHA-665752 | YSK4 | 78.0 | nM |
PHA-665752 | MAP4K5 | 79.0 | nM |
PHA-665752 | HIPK1 | 93.0 | nM |
PHA-665752 | FLT3(D835Y) | 96.0 | nM |
PHA-665752 | AXL | 110.0 | nM |
PHA-665752 | HIPK2 | 120.0 | nM |
PHA-665752 | CDK7 | 130.0 | nM |
PHA-665752 | FLT3(D835H) | 140.0 | nM |
PHA-665752 | M4K1 | 150.0 | nM |
PHA-665752 | MINK | 250.0 | nM |
PHA-665752 | FLT3 | 250.0 | nM |
PHA-665752 | FLT3(K663Q) | 270.0 | nM |
PHA-665752 | PIP5K1A | 280.0 | nM |