PHA-665752 KINOMEscan - Dataset (ID:20166)

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Small Molecule Protein Kd Conc unit
PHA-665752 FES
nM
PHA-665752 FGFR1
nM
PHA-665752 FGFR2 5200.0
nM
PHA-665752 FGFR3 5200.0
nM
PHA-665752 FGFR3(G697C)
nM
PHA-665752 FGFR4
nM
PHA-665752 FGR 1900.0
nM
PHA-665752 VGFR1
nM
PHA-665752 FLT3 250.0
nM
PHA-665752 FLT3(D835H) 140.0
nM
PHA-665752 FLT3(D835Y) 96.0
nM
PHA-665752 FLT3(ITD) 58.0
nM
PHA-665752 FLT3(K663Q) 270.0
nM
PHA-665752 FLT3(N841I) 470.0
nM
PHA-665752 FLT3(R834Q) 4600.0
nM
PHA-665752 FLT4 1400.0
nM
PHA-665752 FRK
nM
PHA-665752 FYN
nM
PHA-665752 GAK 1300.0
nM
PHA-665752 GCN2(Kin.Dom.2,S808G) 3400.0
nM
PHA-665752 GRK1 1100.0
nM
PHA-665752 GRK4 420.0
nM
PHA-665752 GRK7 61.0
nM
PHA-665752 GSK3A
nM
PHA-665752 GSK3B
nM