PHA-665752 KINOMEscan - Dataset (ID:20166)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PHA-665752 | IKKB | nM | |
PHA-665752 | IKKE | 700.0 | nM |
PHA-665752 | INSR | 2300.0 | nM |
PHA-665752 | INSRR | 3500.0 | nM |
PHA-665752 | IRAK1 | 1600.0 | nM |
PHA-665752 | IRAK3 | 610.0 | nM |
PHA-665752 | IRAK4 | 2500.0 | nM |
PHA-665752 | ITK | nM | |
PHA-665752 | JAK1(JH1domain-catalytic) | nM | |
PHA-665752 | JAK1(JH2domain-pseudokinase) | 2700.0 | nM |
PHA-665752 | JAK2(JH1domain-catalytic) | 430.0 | nM |
PHA-665752 | JAK3(JH1domain-catalytic) | 470.0 | nM |
PHA-665752 | JNK1 | nM | |
PHA-665752 | JNK3 | nM | |
PHA-665752 | KC1G1 | nM | |
PHA-665752 | KC1G2 | nM | |
PHA-665752 | KCC2D | 2900.0 | nM |
PHA-665752 | KCC4 | nM | |
PHA-665752 | KGP1 | nM | |
PHA-665752 | KGP2 | nM | |
PHA-665752 | KIT | 3200.0 | nM |
PHA-665752 | KIT(A829P) | 4300.0 | nM |
PHA-665752 | KIT(D816H) | 4000.0 | nM |
PHA-665752 | KIT(D816V) | 590.0 | nM |
PHA-665752 | KIT(L576P) | 1300.0 | nM |