PHA-665752 KINOMEscan - Dataset (ID:20166)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PHA-665752 | FLT3(D835H) | 140.0 | nM |
PHA-665752 | FLT3(D835Y) | 96.0 | nM |
PHA-665752 | FLT3(ITD) | 58.0 | nM |
PHA-665752 | FLT3(K663Q) | 270.0 | nM |
PHA-665752 | FLT3(N841I) | 470.0 | nM |
PHA-665752 | FLT3(R834Q) | 4600.0 | nM |
PHA-665752 | FLT4 | 1400.0 | nM |
PHA-665752 | FRK | nM | |
PHA-665752 | FYN | nM | |
PHA-665752 | GAK | 1300.0 | nM |
PHA-665752 | GCN2(Kin.Dom.2,S808G) | 3400.0 | nM |
PHA-665752 | GRK1 | 1100.0 | nM |
PHA-665752 | GRK4 | 420.0 | nM |
PHA-665752 | GRK7 | 61.0 | nM |
PHA-665752 | GSK3A | nM | |
PHA-665752 | GSK3B | nM | |
PHA-665752 | HCK | nM | |
PHA-665752 | HIPK1 | 93.0 | nM |
PHA-665752 | HIPK2 | 120.0 | nM |
PHA-665752 | HIPK3 | 63.0 | nM |
PHA-665752 | HIPK4 | 1300.0 | nM |
PHA-665752 | HUNK | 1400.0 | nM |
PHA-665752 | ICK | 400.0 | nM |
PHA-665752 | IGF1R | nM | |
PHA-665752 | IKKA | nM |