PHA-665752 KINOMEscan - Dataset (ID:20166)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PHA-665752 | CSNK1D | 4200.0 | nM |
PHA-665752 | S6K1 | 4100.0 | nM |
PHA-665752 | KIT(D816H) | 4000.0 | nM |
PHA-665752 | DRAK1 | 4000.0 | nM |
PHA-665752 | EPHA8 | 3900.0 | nM |
PHA-665752 | ABL1(T315I)-phosphorylated | 3900.0 | nM |
PHA-665752 | ABL1(T315I)-nonphosphorylated | 3800.0 | nM |
PHA-665752 | MST4 | 3800.0 | nM |
PHA-665752 | CLK3 | 3600.0 | nM |
PHA-665752 | MARK2 | 3600.0 | nM |
PHA-665752 | MAP4K2 | 3600.0 | nM |
PHA-665752 | INSRR | 3500.0 | nM |
PHA-665752 | DRAK2 | 3500.0 | nM |
PHA-665752 | GCN2(Kin.Dom.2,S808G) | 3400.0 | nM |
PHA-665752 | CAMK2A | 3400.0 | nM |
PHA-665752 | KIT | 3200.0 | nM |
PHA-665752 | M3K13 | 3200.0 | nM |
PHA-665752 | ROS1 | 3000.0 | nM |
PHA-665752 | ABL1(F317L)-phosphorylated | 2900.0 | nM |
PHA-665752 | PAK1 | 2900.0 | nM |
PHA-665752 | KCC2D | 2900.0 | nM |
PHA-665752 | EPHB6 | 2900.0 | nM |
PHA-665752 | ALK | 2700.0 | nM |
PHA-665752 | JAK1(JH2domain-pseudokinase) | 2700.0 | nM |
PHA-665752 | ABL1-nonphosphorylated | 2600.0 | nM |