PHA-665752 KINOMEscan - Dataset (ID:20166)

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Small Molecule Protein Kd Conc unit
PHA-665752 CSNK1D 4200.0
nM
PHA-665752 S6K1 4100.0
nM
PHA-665752 KIT(D816H) 4000.0
nM
PHA-665752 DRAK1 4000.0
nM
PHA-665752 EPHA8 3900.0
nM
PHA-665752 ABL1(T315I)-phosphorylated 3900.0
nM
PHA-665752 ABL1(T315I)-nonphosphorylated 3800.0
nM
PHA-665752 MST4 3800.0
nM
PHA-665752 CLK3 3600.0
nM
PHA-665752 MARK2 3600.0
nM
PHA-665752 MAP4K2 3600.0
nM
PHA-665752 INSRR 3500.0
nM
PHA-665752 DRAK2 3500.0
nM
PHA-665752 GCN2(Kin.Dom.2,S808G) 3400.0
nM
PHA-665752 CAMK2A 3400.0
nM
PHA-665752 KIT 3200.0
nM
PHA-665752 M3K13 3200.0
nM
PHA-665752 ROS1 3000.0
nM
PHA-665752 ABL1(F317L)-phosphorylated 2900.0
nM
PHA-665752 PAK1 2900.0
nM
PHA-665752 KCC2D 2900.0
nM
PHA-665752 EPHB6 2900.0
nM
PHA-665752 ALK 2700.0
nM
PHA-665752 JAK1(JH2domain-pseudokinase) 2700.0
nM
PHA-665752 ABL1-nonphosphorylated 2600.0
nM