PHA-665752 KINOMEscan - Dataset (ID:20166)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PHA-665752 | RSK2(Kin.Dom.1-N-terminal) | 9900.0 | nM |
PHA-665752 | ABL1(Q252H)-phosphorylated | 9300.0 | nM |
PHA-665752 | ABL1(H396P)-phosphorylated | 9000.0 | nM |
PHA-665752 | NIM1 | 8700.0 | nM |
PHA-665752 | ROCK2 | 8700.0 | nM |
PHA-665752 | PLK2 | 8300.0 | nM |
PHA-665752 | ABL1-phosphorylated | 8200.0 | nM |
PHA-665752 | MYLK | 7900.0 | nM |
PHA-665752 | DDR2 | 7600.0 | nM |
PHA-665752 | KIT(V559D,V654A) | 7200.0 | nM |
PHA-665752 | ABL2 | 6900.0 | nM |
PHA-665752 | RSK4(Kin.Dom.1-N-terminal) | 6800.0 | nM |
PHA-665752 | TIE2 | 6700.0 | nM |
PHA-665752 | TYK2(JH2domain-pseudokinase) | 6600.0 | nM |
PHA-665752 | BMPR2 | 6200.0 | nM |
PHA-665752 | MAP3K3 | 5900.0 | nM |
PHA-665752 | CSNK2A2 | 5600.0 | nM |
PHA-665752 | TAK1 | 5300.0 | nM |
PHA-665752 | M3K2 | 5200.0 | nM |
PHA-665752 | FGFR3 | 5200.0 | nM |
PHA-665752 | FGFR2 | 5200.0 | nM |
PHA-665752 | STK16 | 4800.0 | nM |
PHA-665752 | FLT3(R834Q) | 4600.0 | nM |
PHA-665752 | DCAMKL3 | 4500.0 | nM |
PHA-665752 | KIT(A829P) | 4300.0 | nM |