PHA-665752 KINOMEscan - Dataset (ID:20166)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
PHA-665752 | KIT | 3200.0 | nM |
PHA-665752 | KIT(A829P) | 4300.0 | nM |
PHA-665752 | KIT(D816H) | 4000.0 | nM |
PHA-665752 | KIT(D816V) | 590.0 | nM |
PHA-665752 | KIT(L576P) | 1300.0 | nM |
PHA-665752 | KIT(V559D) | 2500.0 | nM |
PHA-665752 | KIT(V559D,T670I) | nM | |
PHA-665752 | KIT(V559D,V654A) | 7200.0 | nM |
PHA-665752 | LATS1 | nM | |
PHA-665752 | LATS2 | nM | |
PHA-665752 | LCK | 320.0 | nM |
PHA-665752 | LIMK1 | nM | |
PHA-665752 | LIMK2 | nM | |
PHA-665752 | LKB1 | 2600.0 | nM |
PHA-665752 | LOK | 290.0 | nM |
PHA-665752 | LRRK2 | nM | |
PHA-665752 | LRRK2(G2019S) | nM | |
PHA-665752 | LTK | nM | |
PHA-665752 | LYN | nM | |
PHA-665752 | M3K13 | 3200.0 | nM |
PHA-665752 | MAK | 890.0 | nM |
PHA-665752 | MAP3K1 | nM | |
PHA-665752 | MAP3K15 | nM | |
PHA-665752 | M3K2 | 5200.0 | nM |
PHA-665752 | MAP3K3 | 5900.0 | nM |