SGX-523 KINOMEscan - Dataset (ID:20165)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
SGX523 | MET | 0.2 | nM |
SGX523 | MET(M1250T) | 0.8 | nM |
SGX523 | MET(Y1235D) | 3.9 | nM |
SGX523 | DYRK1A | 780.0 | nM |
SGX523 | DYRK1B | 1800.0 | nM |
SGX523 | JNK3 | 1900.0 | nM |
SGX523 | PI42C | 3300.0 | nM |
SGX523 | ABL1(H396P)-nonphosphorylated | 3400.0 | nM |
SGX523 | JNK1 | 4200.0 | nM |
SGX523 | YSK4 | 6400.0 | nM |
SGX523 | ABL1(Y253F)-phosphorylated | nM | |
SGX523 | ABL1(T315I)-phosphorylated | nM | |
SGX523 | ABL1(T315I)-nonphosphorylated | nM | |
SGX523 | ABL1-nonphosphorylated | nM | |
SGX523 | ABL1(F317L)-phosphorylated | nM | |
SGX523 | ABL1(F317I)-nonphosphorylated | nM | |
SGX523 | ABL1(Q252H)-phosphorylated | nM | |
SGX523 | ACVR2B | nM | |
SGX523 | ACVR2A | nM | |
SGX523 | ABL1(Q252H)-nonphosphorylated | nM | |
SGX523 | ACVRL1 | nM | |
SGX523 | ADCK3 | nM | |
SGX523 | ADCK4 | nM | |
SGX523 | ABL1(F317L)-nonphosphorylated | nM | |
SGX523 | ACVR1B | nM |