Pazopanib KINOMEscan - Dataset (ID:20163)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pazopanib | IKKB | nM | |
Pazopanib | IKKE | nM | |
Pazopanib | INSR | nM | |
Pazopanib | INSRR | nM | |
Pazopanib | IRAK1 | 5900.0 | nM |
Pazopanib | IRAK3 | 800.0 | nM |
Pazopanib | IRAK4 | nM | |
Pazopanib | ITK | nM | |
Pazopanib | JAK1(JH1domain-catalytic) | nM | |
Pazopanib | JAK1(JH2domain-pseudokinase) | nM | |
Pazopanib | JAK2(JH1domain-catalytic) | 1700.0 | nM |
Pazopanib | JAK3(JH1domain-catalytic) | 6900.0 | nM |
Pazopanib | JNK1 | 2000.0 | nM |
Pazopanib | JNK3 | 1900.0 | nM |
Pazopanib | KC1G1 | nM | |
Pazopanib | KC1G2 | nM | |
Pazopanib | KCC2D | nM | |
Pazopanib | KCC4 | nM | |
Pazopanib | KGP1 | nM | |
Pazopanib | KGP2 | nM | |
Pazopanib | KIT | 2.8 | nM |
Pazopanib | KIT(A829P) | 33.0 | nM |
Pazopanib | KIT(D816H) | 1000.0 | nM |
Pazopanib | KIT(D816V) | 500.0 | nM |
Pazopanib | KIT(L576P) | 1.8 | nM |