Pazopanib KINOMEscan - Dataset (ID:20163)

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Small Molecule Protein Kd Conc unit
Pazopanib LIMK1 720.0
nM
Pazopanib BRAF 730.0
nM
Pazopanib MLK3 740.0
nM
Pazopanib FLT3(K663Q) 740.0
nM
Pazopanib FGFR3 740.0
nM
Pazopanib M4K1 750.0
nM
Pazopanib FRK 750.0
nM
Pazopanib AURKC 750.0
nM
Pazopanib IRAK3 800.0
nM
Pazopanib ABL1(E255K)-phosphorylated 800.0
nM
Pazopanib FLT3(D835Y) 810.0
nM
Pazopanib RAF1 900.0
nM
Pazopanib ROS1 920.0
nM
Pazopanib YSK4 940.0
nM
Pazopanib PIK4CB 960.0
nM
Pazopanib NEK2 980.0
nM
Pazopanib FGFR1 990.0
nM
Pazopanib KIT(D816H) 1000.0
nM
Pazopanib BMPR1B 1000.0
nM
Pazopanib FLT3(D835H) 1100.0
nM
Pazopanib FLT3 1100.0
nM
Pazopanib LYN 1100.0
nM
Pazopanib LCK 1200.0
nM
Pazopanib CDK16 1200.0
nM
Pazopanib CDC2L2 1300.0
nM