Pazopanib KINOMEscan - Dataset (ID:20163)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pazopanib | PLK4 | 290.0 | nM |
Pazopanib | M3K2 | 290.0 | nM |
Pazopanib | MLK1 | 290.0 | nM |
Pazopanib | TNIK | 310.0 | nM |
Pazopanib | RET | 310.0 | nM |
Pazopanib | STK16 | 360.0 | nM |
Pazopanib | PFCDPK1(P.falciparum) | 370.0 | nM |
Pazopanib | ABL1(H396P)-nonphosphorylated | 380.0 | nM |
Pazopanib | LIMK2 | 390.0 | nM |
Pazopanib | BRAF(V600E) | 430.0 | nM |
Pazopanib | STK36 | 470.0 | nM |
Pazopanib | ABL1(Y253F)-phosphorylated | 480.0 | nM |
Pazopanib | MP2K5 | 480.0 | nM |
Pazopanib | KIT(D816V) | 500.0 | nM |
Pazopanib | ABL1(Q252H)-phosphorylated | 530.0 | nM |
Pazopanib | ABL1(Q252H)-nonphosphorylated | 530.0 | nM |
Pazopanib | ABL1(M351T)-phosphorylated | 560.0 | nM |
Pazopanib | RIPK2 | 580.0 | nM |
Pazopanib | MP2K4 | 590.0 | nM |
Pazopanib | RIOK2 | 610.0 | nM |
Pazopanib | ABL1-nonphosphorylated | 620.0 | nM |
Pazopanib | FGFR3(G697C) | 620.0 | nM |
Pazopanib | ABL1-phosphorylated | 650.0 | nM |
Pazopanib | TIE1 | 700.0 | nM |
Pazopanib | ABL1(H396P)-phosphorylated | 700.0 | nM |