Pazopanib KINOMEscan - Dataset (ID:20163)

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Small Molecule Protein Kd Conc unit
Pazopanib KIT 2.8
nM
Pazopanib KIT(A829P) 33.0
nM
Pazopanib KIT(D816H) 1000.0
nM
Pazopanib KIT(D816V) 500.0
nM
Pazopanib KIT(L576P) 1.8
nM
Pazopanib KIT(V559D) 2.3
nM
Pazopanib KIT(V559D,T670I) 6.5
nM
Pazopanib KIT(V559D,V654A) 30.0
nM
Pazopanib LATS1
nM
Pazopanib LATS2
nM
Pazopanib LCK 1200.0
nM
Pazopanib LIMK1 720.0
nM
Pazopanib LIMK2 390.0
nM
Pazopanib LKB1
nM
Pazopanib LOK 84.0
nM
Pazopanib LRRK2
nM
Pazopanib LRRK2(G2019S)
nM
Pazopanib LTK 6800.0
nM
Pazopanib LYN 1100.0
nM
Pazopanib M3K13
nM
Pazopanib MAK
nM
Pazopanib MAP3K1 2900.0
nM
Pazopanib MAP3K15
nM
Pazopanib M3K2 290.0
nM
Pazopanib MAP3K3
nM