Pazopanib KINOMEscan - Dataset (ID:20163)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Pazopanib | FES | 1400.0 | nM |
Pazopanib | FGFR1 | 990.0 | nM |
Pazopanib | FGFR2 | 210.0 | nM |
Pazopanib | FGFR3 | 740.0 | nM |
Pazopanib | FGFR3(G697C) | 620.0 | nM |
Pazopanib | FGFR4 | 2800.0 | nM |
Pazopanib | FGR | 1600.0 | nM |
Pazopanib | VGFR1 | 14.0 | nM |
Pazopanib | FLT3 | 1100.0 | nM |
Pazopanib | FLT3(D835H) | 1100.0 | nM |
Pazopanib | FLT3(D835Y) | 810.0 | nM |
Pazopanib | FLT3(ITD) | 2500.0 | nM |
Pazopanib | FLT3(K663Q) | 740.0 | nM |
Pazopanib | FLT3(N841I) | 1600.0 | nM |
Pazopanib | FLT3(R834Q) | 9600.0 | nM |
Pazopanib | FLT4 | 27.0 | nM |
Pazopanib | FRK | 750.0 | nM |
Pazopanib | FYN | 2700.0 | nM |
Pazopanib | GAK | 200.0 | nM |
Pazopanib | GCN2(Kin.Dom.2,S808G) | nM | |
Pazopanib | GRK1 | nM | |
Pazopanib | GRK4 | nM | |
Pazopanib | GRK7 | nM | |
Pazopanib | GSK3A | nM | |
Pazopanib | GSK3B | nM |