Pazopanib KINOMEscan - Dataset (ID:20163)

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Small Molecule Protein Kd Conc unit
Pazopanib FES 1400.0
nM
Pazopanib FGFR1 990.0
nM
Pazopanib FGFR2 210.0
nM
Pazopanib FGFR3 740.0
nM
Pazopanib FGFR3(G697C) 620.0
nM
Pazopanib FGFR4 2800.0
nM
Pazopanib FGR 1600.0
nM
Pazopanib VGFR1 14.0
nM
Pazopanib FLT3 1100.0
nM
Pazopanib FLT3(D835H) 1100.0
nM
Pazopanib FLT3(D835Y) 810.0
nM
Pazopanib FLT3(ITD) 2500.0
nM
Pazopanib FLT3(K663Q) 740.0
nM
Pazopanib FLT3(N841I) 1600.0
nM
Pazopanib FLT3(R834Q) 9600.0
nM
Pazopanib FLT4 27.0
nM
Pazopanib FRK 750.0
nM
Pazopanib FYN 2700.0
nM
Pazopanib GAK 200.0
nM
Pazopanib GCN2(Kin.Dom.2,S808G)
nM
Pazopanib GRK1
nM
Pazopanib GRK4
nM
Pazopanib GRK7
nM
Pazopanib GSK3A
nM
Pazopanib GSK3B
nM