Nilotinib KINOMEscan - Dataset (ID:20162)

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Small Molecule Protein Kd Conc unit
Nilotinib PGFRB 73.0
nM
Nilotinib FRK 86.0
nM
Nilotinib LYN 100.0
nM
Nilotinib EPHA3 110.0
nM
Nilotinib KIT(V559D,T670I) 150.0
nM
Nilotinib PGFRA 180.0
nM
Nilotinib MP2K5 190.0
nM
Nilotinib EPHA2 230.0
nM
Nilotinib KIT(V559D,V654A) 260.0
nM
Nilotinib FGR 320.0
nM
Nilotinib EPHA4 330.0
nM
Nilotinib TNNI3K 360.0
nM
Nilotinib HCK 390.0
nM
Nilotinib JNK1 450.0
nM
Nilotinib MK14 460.0
nM
Nilotinib TRKB 490.0
nM
Nilotinib BLK 500.0
nM
Nilotinib EPHB6 500.0
nM
Nilotinib KIT(D816H) 540.0
nM
Nilotinib BRAF(V600E) 570.0
nM
Nilotinib EPHA1 590.0
nM
Nilotinib TRKC 600.0
nM
Nilotinib EPHB2 640.0
nM
Nilotinib EPHA6 640.0
nM
Nilotinib ABL1(T315I)-nonphosphorylated 660.0
nM