Nilotinib KINOMEscan - Dataset (ID:20162)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Nilotinib | PGFRB | 73.0 | nM |
Nilotinib | FRK | 86.0 | nM |
Nilotinib | LYN | 100.0 | nM |
Nilotinib | EPHA3 | 110.0 | nM |
Nilotinib | KIT(V559D,T670I) | 150.0 | nM |
Nilotinib | PGFRA | 180.0 | nM |
Nilotinib | MP2K5 | 190.0 | nM |
Nilotinib | EPHA2 | 230.0 | nM |
Nilotinib | KIT(V559D,V654A) | 260.0 | nM |
Nilotinib | FGR | 320.0 | nM |
Nilotinib | EPHA4 | 330.0 | nM |
Nilotinib | TNNI3K | 360.0 | nM |
Nilotinib | HCK | 390.0 | nM |
Nilotinib | JNK1 | 450.0 | nM |
Nilotinib | MK14 | 460.0 | nM |
Nilotinib | TRKB | 490.0 | nM |
Nilotinib | BLK | 500.0 | nM |
Nilotinib | EPHB6 | 500.0 | nM |
Nilotinib | KIT(D816H) | 540.0 | nM |
Nilotinib | BRAF(V600E) | 570.0 | nM |
Nilotinib | EPHA1 | 590.0 | nM |
Nilotinib | TRKC | 600.0 | nM |
Nilotinib | EPHB2 | 640.0 | nM |
Nilotinib | EPHA6 | 640.0 | nM |
Nilotinib | ABL1(T315I)-nonphosphorylated | 660.0 | nM |