Nilotinib KINOMEscan - Dataset (ID:20162)
Proteins Studied
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LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200451 | TYK2(JH2domain-pseudokinase) | 200451 | P29597 | Non-receptor tyrosine-protein kinase TYK2; Tyrosine kinase 2; JTK1; TYK2 | KINOMEscan | JH2domain-pseudokinase | Wild Type; Partial length | ||
200454 | TYRO3 | 200454 | Q06418 | TYRO3 protein tyrosine kinase; BYK; Dtk; FLJ16467; RSE; Sky; Tif; TYRO3; Tyro3/Sky | KINOMEscan | Wild Type; Partial length | |||
200025 | ABL1-phosphorylated | 200025 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | phosphorylated | Wild Type; Partial length | ||
200013 | ABL1(H396P)-phosphorylated | 200013 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | H396P | phosphorylated | Mutation (H396P); Partial length | |
200015 | ABL1(M351T)-phosphorylated | 200015 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | M351T | phosphorylated | Mutation (M351T); Partial length | |
200018 | ABL1(Q252H)-phosphorylated | 200018 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | Q252H | phosphorylated | Mutation (Q252H); Partial length | |
200021 | ABL1(T315I)-phosphorylated | 200021 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | T315I | phosphorylated | Mutation (T315I); Partial length | |
200023 | ABL1(Y253F)-phosphorylated | 200023 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | Y253F | phosphorylated | Mutation (Y253F); Partial length | |
200004 | ABL1(E255K)-phosphorylated | 200004 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | E255K | phosphorylated | Mutation (E255K); Partial length | |
200007 | ABL1(F317I)-phosphorylated | 200007 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | F317I | phosphorylated | Mutation (F317I); Partial length | |
200010 | ABL1(F317L)-phosphorylated | 200010 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | F317L | phosphorylated | Mutation (F317L); Partial length | |
200006 | ABL1(F317I)-nonphosphorylated | 200006 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | F317I | nonphosphorylated | Mutation (F317I); Partial length | |
200020 | ABL1(T315I)-nonphosphorylated | 200020 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | T315I | nonphosphorylated | Mutation (T315I); Partial length | |
200009 | ABL1(F317L)-nonphosphorylated | 200009 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | F317L | nonphosphorylated | Mutation (F317L); Partial length | |
200017 | ABL1(Q252H)-nonphosphorylated | 200017 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | Q252H | nonphosphorylated | Mutation (Q252H); Partial length | |
200012 | ABL1(H396P)-nonphosphorylated | 200012 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | H396P | nonphosphorylated | Mutation (H396P); Partial length | |
200024 | ABL1-nonphosphorylated | 200024 | P00519 | C-abl oncogene 1, receptor tyrosine kinase; ABL; ABL1; bcr/abl; c-ABL; JTK7; p150; v-abl | KINOMEscan | nonphosphorylated | Wild Type; Partial length |