Gefitinib KINOMEscan - Dataset (ID:20161)

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Small Molecule Protein Kd Conc unit
Gefitinib KIT
nM
Gefitinib KIT(A829P) 1800.0
nM
Gefitinib KIT(D816H) 5500.0
nM
Gefitinib KIT(D816V) 4300.0
nM
Gefitinib KIT(L576P)
nM
Gefitinib KIT(V559D)
nM
Gefitinib KIT(V559D,T670I)
nM
Gefitinib KIT(V559D,V654A)
nM
Gefitinib LATS1
nM
Gefitinib LATS2
nM
Gefitinib LCK 630.0
nM
Gefitinib LIMK1
nM
Gefitinib LIMK2
nM
Gefitinib LKB1
nM
Gefitinib LOK 470.0
nM
Gefitinib LRRK2
nM
Gefitinib LRRK2(G2019S)
nM
Gefitinib LTK 5500.0
nM
Gefitinib LYN 990.0
nM
Gefitinib M3K13
nM
Gefitinib MAK
nM
Gefitinib MAP3K1
nM
Gefitinib MAP3K15
nM
Gefitinib M3K2 3300.0
nM
Gefitinib MAP3K3 2100.0
nM