Gefitinib KINOMEscan - Dataset (ID:20161)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Gefitinib | KIT | nM | |
Gefitinib | KIT(A829P) | 1800.0 | nM |
Gefitinib | KIT(D816H) | 5500.0 | nM |
Gefitinib | KIT(D816V) | 4300.0 | nM |
Gefitinib | KIT(L576P) | nM | |
Gefitinib | KIT(V559D) | nM | |
Gefitinib | KIT(V559D,T670I) | nM | |
Gefitinib | KIT(V559D,V654A) | nM | |
Gefitinib | LATS1 | nM | |
Gefitinib | LATS2 | nM | |
Gefitinib | LCK | 630.0 | nM |
Gefitinib | LIMK1 | nM | |
Gefitinib | LIMK2 | nM | |
Gefitinib | LKB1 | nM | |
Gefitinib | LOK | 470.0 | nM |
Gefitinib | LRRK2 | nM | |
Gefitinib | LRRK2(G2019S) | nM | |
Gefitinib | LTK | 5500.0 | nM |
Gefitinib | LYN | 990.0 | nM |
Gefitinib | M3K13 | nM | |
Gefitinib | MAK | nM | |
Gefitinib | MAP3K1 | nM | |
Gefitinib | MAP3K15 | nM | |
Gefitinib | M3K2 | 3300.0 | nM |
Gefitinib | MAP3K3 | 2100.0 | nM |