Gefitinib KINOMEscan - Dataset (ID:20161)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Gefitinib | ABL1(M351T)-phosphorylated | 520.0 | nM |
| Gefitinib | RIPK2 | 530.0 | nM |
| Gefitinib | IRAK4 | 540.0 | nM |
| Gefitinib | SBK1 | 560.0 | nM |
| Gefitinib | EPHA6 | 590.0 | nM |
| Gefitinib | MP2K5 | 600.0 | nM |
| Gefitinib | CDK7 | 610.0 | nM |
| Gefitinib | LCK | 630.0 | nM |
| Gefitinib | ABL1(H396P)-nonphosphorylated | 680.0 | nM |
| Gefitinib | ABL1(F317L)-phosphorylated | 780.0 | nM |
| Gefitinib | ERBB3 | 790.0 | nM |
| Gefitinib | CHK2 | 800.0 | nM |
| Gefitinib | SLK | 920.0 | nM |
| Gefitinib | LYN | 990.0 | nM |
| Gefitinib | FLT3(D835Y) | 1000.0 | nM |
| Gefitinib | FLT3(D835H) | 1100.0 | nM |
| Gefitinib | ABL1(Q252H)-nonphosphorylated | 1100.0 | nM |
| Gefitinib | RPS6KA4(Kin.Dom.2-C-terminal) | 1200.0 | nM |
| Gefitinib | MKNK2 | 1200.0 | nM |
| Gefitinib | BLK | 1200.0 | nM |
| Gefitinib | EPHB1 | 1300.0 | nM |
| Gefitinib | CIT | 1300.0 | nM |
| Gefitinib | EPHA5 | 1500.0 | nM |
| Gefitinib | IRAK3 | 1500.0 | nM |
| Gefitinib | ABL2 | 1600.0 | nM |