Gefitinib KINOMEscan - Dataset (ID:20161)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Gefitinib | PI42C | 7500.0 | nM |
Gefitinib | DMPK | 6900.0 | nM |
Gefitinib | TNIK | 6900.0 | nM |
Gefitinib | TXK | 6000.0 | nM |
Gefitinib | PIM3 | 5800.0 | nM |
Gefitinib | STK36 | 5700.0 | nM |
Gefitinib | DAPK3 | 5700.0 | nM |
Gefitinib | LTK | 5500.0 | nM |
Gefitinib | KIT(D816H) | 5500.0 | nM |
Gefitinib | EPHA3 | 5500.0 | nM |
Gefitinib | FLT3(K663Q) | 5100.0 | nM |
Gefitinib | ABL1(F317I)-phosphorylated | 4700.0 | nM |
Gefitinib | SNARK | 4600.0 | nM |
Gefitinib | HCK | 4400.0 | nM |
Gefitinib | KIT(D816V) | 4300.0 | nM |
Gefitinib | NLK | 4200.0 | nM |
Gefitinib | EPHA1 | 4000.0 | nM |
Gefitinib | SRC | 3800.0 | nM |
Gefitinib | DRAK2 | 3800.0 | nM |
Gefitinib | PHKG1 | 3700.0 | nM |
Gefitinib | FLT3(R834Q) | 3500.0 | nM |
Gefitinib | KPCD1 | 3500.0 | nM |
Gefitinib | MET(Y1235D) | 3500.0 | nM |
Gefitinib | ERBB2 | 3500.0 | nM |
Gefitinib | M3K2 | 3300.0 | nM |