LY-317615 KINOMEscan - Dataset (ID:20159)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Enzastaurin | FES | nM | |
| Enzastaurin | FGFR1 | 4000.0 | nM |
| Enzastaurin | FGFR2 | nM | |
| Enzastaurin | FGFR3 | nM | |
| Enzastaurin | FGFR3(G697C) | nM | |
| Enzastaurin | FGFR4 | nM | |
| Enzastaurin | FGR | nM | |
| Enzastaurin | VGFR1 | nM | |
| Enzastaurin | FLT3 | 330.0 | nM |
| Enzastaurin | FLT3(D835H) | 49.0 | nM |
| Enzastaurin | FLT3(D835Y) | 40.0 | nM |
| Enzastaurin | FLT3(ITD) | 72.0 | nM |
| Enzastaurin | FLT3(K663Q) | 420.0 | nM |
| Enzastaurin | FLT3(N841I) | 250.0 | nM |
| Enzastaurin | FLT3(R834Q) | 1800.0 | nM |
| Enzastaurin | FLT4 | 3800.0 | nM |
| Enzastaurin | FRK | nM | |
| Enzastaurin | FYN | nM | |
| Enzastaurin | GAK | nM | |
| Enzastaurin | GCN2(Kin.Dom.2,S808G) | nM | |
| Enzastaurin | GRK1 | 1700.0 | nM |
| Enzastaurin | GRK4 | nM | |
| Enzastaurin | GRK7 | 1300.0 | nM |
| Enzastaurin | GSK3A | nM | |
| Enzastaurin | GSK3B | 8.3 | nM |