LY-317615 KINOMEscan - Dataset (ID:20159)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Enzastaurin | PRKX | nM | |
Enzastaurin | PRP4 | nM | |
Enzastaurin | FAK2 | nM | |
Enzastaurin | SIK3 | nM | |
Enzastaurin | RAF1 | nM | |
Enzastaurin | RET | nM | |
Enzastaurin | RET(M918T) | nM | |
Enzastaurin | RET(V804L) | nM | |
Enzastaurin | RET(V804M) | nM | |
Enzastaurin | RIOK1 | nM | |
Enzastaurin | RIOK2 | nM | |
Enzastaurin | RIOK3 | nM | |
Enzastaurin | RIPK1 | nM | |
Enzastaurin | RIPK2 | nM | |
Enzastaurin | RIPK4 | nM | |
Enzastaurin | RIPK5 | nM | |
Enzastaurin | ROCK1 | nM | |
Enzastaurin | ROCK2 | nM | |
Enzastaurin | ROS1 | nM | |
Enzastaurin | RPS6KA4(Kin.Dom.1-N-terminal) | 2500.0 | nM |
Enzastaurin | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
Enzastaurin | RPS6KA5(Kin.Dom.1-N-terminal) | 370.0 | nM |
Enzastaurin | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
Enzastaurin | RSK1(Kin.Dom.1-N-terminal) | 1600.0 | nM |
Enzastaurin | RSK1(Kin.Dom.2-C-terminal) | nM |