LY-317615 KINOMEscan - Dataset (ID:20159)

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Small Molecule Protein Kd Conc unit
Enzastaurin ICK 680.0
nM
Enzastaurin HIPK2 720.0
nM
Enzastaurin DRAK1 760.0
nM
Enzastaurin PIM2 870.0
nM
Enzastaurin AKT3 1000.0
nM
Enzastaurin DYRK1B 1000.0
nM
Enzastaurin HIPK1 1000.0
nM
Enzastaurin KIT(D816V) 1100.0
nM
Enzastaurin KGP1 1100.0
nM
Enzastaurin CDK3 1100.0
nM
Enzastaurin PIM3 1100.0
nM
Enzastaurin HIPK4 1200.0
nM
Enzastaurin GRK7 1300.0
nM
Enzastaurin CDK9 1300.0
nM
Enzastaurin TLK2 1400.0
nM
Enzastaurin CDK14 1500.0
nM
Enzastaurin YSK4 1600.0
nM
Enzastaurin RSK1(Kin.Dom.1-N-terminal) 1600.0
nM
Enzastaurin CLK4 1600.0
nM
Enzastaurin JAK3(JH1domain-catalytic) 1700.0
nM
Enzastaurin GRK1 1700.0
nM
Enzastaurin M4K1 1800.0
nM
Enzastaurin S6K1 1800.0
nM
Enzastaurin FLT3(R834Q) 1800.0
nM
Enzastaurin MST2 1900.0
nM