LY-317615 KINOMEscan - Dataset (ID:20159)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Enzastaurin | ICK | 680.0 | nM |
Enzastaurin | HIPK2 | 720.0 | nM |
Enzastaurin | DRAK1 | 760.0 | nM |
Enzastaurin | PIM2 | 870.0 | nM |
Enzastaurin | AKT3 | 1000.0 | nM |
Enzastaurin | DYRK1B | 1000.0 | nM |
Enzastaurin | HIPK1 | 1000.0 | nM |
Enzastaurin | KIT(D816V) | 1100.0 | nM |
Enzastaurin | KGP1 | 1100.0 | nM |
Enzastaurin | CDK3 | 1100.0 | nM |
Enzastaurin | PIM3 | 1100.0 | nM |
Enzastaurin | HIPK4 | 1200.0 | nM |
Enzastaurin | GRK7 | 1300.0 | nM |
Enzastaurin | CDK9 | 1300.0 | nM |
Enzastaurin | TLK2 | 1400.0 | nM |
Enzastaurin | CDK14 | 1500.0 | nM |
Enzastaurin | YSK4 | 1600.0 | nM |
Enzastaurin | RSK1(Kin.Dom.1-N-terminal) | 1600.0 | nM |
Enzastaurin | CLK4 | 1600.0 | nM |
Enzastaurin | JAK3(JH1domain-catalytic) | 1700.0 | nM |
Enzastaurin | GRK1 | 1700.0 | nM |
Enzastaurin | M4K1 | 1800.0 | nM |
Enzastaurin | S6K1 | 1800.0 | nM |
Enzastaurin | FLT3(R834Q) | 1800.0 | nM |
Enzastaurin | MST2 | 1900.0 | nM |