MLN-8054 KINOMEscan - Dataset (ID:20157)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
MLN8054 | ROS1 | 3100.0 | nM |
MLN8054 | FLT4 | 3100.0 | nM |
MLN8054 | BMX | 3100.0 | nM |
MLN8054 | EGFR(L858R) | 3200.0 | nM |
MLN8054 | CLK2 | 3200.0 | nM |
MLN8054 | ABL2 | 3300.0 | nM |
MLN8054 | EPHB3 | 3500.0 | nM |
MLN8054 | LOK | 3700.0 | nM |
MLN8054 | BTK | 4200.0 | nM |
MLN8054 | DDR1 | 4200.0 | nM |
MLN8054 | FER | 4400.0 | nM |
MLN8054 | RSK1(Kin.Dom.1-N-terminal) | 4800.0 | nM |
MLN8054 | EGFR(L747-S752del, P753S) | 6400.0 | nM |
MLN8054 | CSK | 9000.0 | nM |
MLN8054 | DAPK2 | 9100.0 | nM |
MLN8054 | FLT3(K663Q) | 9500.0 | nM |
MLN8054 | CDC2L2 | nM | |
MLN8054 | CDC2L1 | nM | |
MLN8054 | ANKK1 | nM | |
MLN8054 | CASK | nM | |
MLN8054 | CAMKK2 | nM | |
MLN8054 | AMPK-alpha2 | nM | |
MLN8054 | KKCC1 | nM | |
MLN8054 | KCC4 | nM | |
MLN8054 | CAMK2G | nM |