MLN-8054 KINOMEscan - Dataset (ID:20157)

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Small Molecule Protein Kd Conc unit
MLN8054 ABL1(Y253F)-phosphorylated 1000.0
nM
MLN8054 VGFR1 1000.0
nM
MLN8054 EPHA7 1000.0
nM
MLN8054 ABL1-nonphosphorylated 1100.0
nM
MLN8054 FGFR3 1200.0
nM
MLN8054 FYN 1300.0
nM
MLN8054 FGFR3(G697C) 1300.0
nM
MLN8054 ABL1(Q252H)-phosphorylated 1300.0
nM
MLN8054 LYN 1400.0
nM
MLN8054 EPHA5 1400.0
nM
MLN8054 IRAK3 1400.0
nM
MLN8054 HCK 1500.0
nM
MLN8054 ABL1(T315I)-nonphosphorylated 1600.0
nM
MLN8054 TIE1 1600.0
nM
MLN8054 FGFR2 1700.0
nM
MLN8054 SIK1 1700.0
nM
MLN8054 EPHA1 1800.0
nM
MLN8054 ABL1(E255K)-phosphorylated 1900.0
nM
MLN8054 FAK2 2000.0
nM
MLN8054 EPHA3 2100.0
nM
MLN8054 CLK3 2300.0
nM
MLN8054 FGFR1 2400.0
nM
MLN8054 TNK1 2400.0
nM
MLN8054 ABL1(T315I)-phosphorylated 2800.0
nM
MLN8054 FLT4 3100.0
nM