MLN-8054 KINOMEscan - Dataset (ID:20157)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
MLN8054 | ABL1(Y253F)-phosphorylated | 1000.0 | nM |
MLN8054 | VGFR1 | 1000.0 | nM |
MLN8054 | EPHA7 | 1000.0 | nM |
MLN8054 | ABL1-nonphosphorylated | 1100.0 | nM |
MLN8054 | FGFR3 | 1200.0 | nM |
MLN8054 | FYN | 1300.0 | nM |
MLN8054 | FGFR3(G697C) | 1300.0 | nM |
MLN8054 | ABL1(Q252H)-phosphorylated | 1300.0 | nM |
MLN8054 | LYN | 1400.0 | nM |
MLN8054 | EPHA5 | 1400.0 | nM |
MLN8054 | IRAK3 | 1400.0 | nM |
MLN8054 | HCK | 1500.0 | nM |
MLN8054 | ABL1(T315I)-nonphosphorylated | 1600.0 | nM |
MLN8054 | TIE1 | 1600.0 | nM |
MLN8054 | FGFR2 | 1700.0 | nM |
MLN8054 | SIK1 | 1700.0 | nM |
MLN8054 | EPHA1 | 1800.0 | nM |
MLN8054 | ABL1(E255K)-phosphorylated | 1900.0 | nM |
MLN8054 | FAK2 | 2000.0 | nM |
MLN8054 | EPHA3 | 2100.0 | nM |
MLN8054 | CLK3 | 2300.0 | nM |
MLN8054 | FGFR1 | 2400.0 | nM |
MLN8054 | TNK1 | 2400.0 | nM |
MLN8054 | ABL1(T315I)-phosphorylated | 2800.0 | nM |
MLN8054 | FLT4 | 3100.0 | nM |