MLN-8054 KINOMEscan - Dataset (ID:20157)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
MLN8054 | FES | nM | |
MLN8054 | FGFR1 | 2400.0 | nM |
MLN8054 | FGFR2 | 1700.0 | nM |
MLN8054 | FGFR3 | 1200.0 | nM |
MLN8054 | FGFR3(G697C) | 1300.0 | nM |
MLN8054 | FGFR4 | nM | |
MLN8054 | FGR | 220.0 | nM |
MLN8054 | VGFR1 | 1000.0 | nM |
MLN8054 | FLT3 | nM | |
MLN8054 | FLT3(D835H) | nM | |
MLN8054 | FLT3(D835Y) | nM | |
MLN8054 | FLT3(ITD) | nM | |
MLN8054 | FLT3(K663Q) | 9500.0 | nM |
MLN8054 | FLT3(N841I) | nM | |
MLN8054 | FLT3(R834Q) | nM | |
MLN8054 | FLT4 | 3100.0 | nM |
MLN8054 | FRK | nM | |
MLN8054 | FYN | 1300.0 | nM |
MLN8054 | GAK | nM | |
MLN8054 | GCN2(Kin.Dom.2,S808G) | nM | |
MLN8054 | GRK1 | nM | |
MLN8054 | GRK4 | nM | |
MLN8054 | GRK7 | nM | |
MLN8054 | GSK3A | nM | |
MLN8054 | GSK3B | nM |