MLN-8054 KINOMEscan - Dataset (ID:20157)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
MLN8054 | PRKX | nM | |
MLN8054 | PRP4 | nM | |
MLN8054 | FAK2 | 2000.0 | nM |
MLN8054 | SIK3 | nM | |
MLN8054 | RAF1 | nM | |
MLN8054 | RET | nM | |
MLN8054 | RET(M918T) | nM | |
MLN8054 | RET(V804L) | nM | |
MLN8054 | RET(V804M) | nM | |
MLN8054 | RIOK1 | nM | |
MLN8054 | RIOK2 | nM | |
MLN8054 | RIOK3 | nM | |
MLN8054 | RIPK1 | nM | |
MLN8054 | RIPK2 | nM | |
MLN8054 | RIPK4 | nM | |
MLN8054 | RIPK5 | nM | |
MLN8054 | ROCK1 | nM | |
MLN8054 | ROCK2 | nM | |
MLN8054 | ROS1 | 3100.0 | nM |
MLN8054 | RPS6KA4(Kin.Dom.1-N-terminal) | nM | |
MLN8054 | RPS6KA4(Kin.Dom.2-C-terminal) | nM | |
MLN8054 | RPS6KA5(Kin.Dom.1-N-terminal) | nM | |
MLN8054 | RPS6KA5(Kin.Dom.2-C-terminal) | nM | |
MLN8054 | RSK1(Kin.Dom.1-N-terminal) | 4800.0 | nM |
MLN8054 | RSK1(Kin.Dom.2-C-terminal) | nM |