MLN-8054 KINOMEscan - Dataset (ID:20157)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200276 MST4 200276 Q9P289
Serine/threonine protein kinase MST4; MASK; MST4
KINOMEscan Wild Type; Full length
200135 EPHA1 200135 P21709
EPH receptor A1; EPH; EPHA1; EPHT; EPHT1; MGC163163
KINOMEscan Wild Type; Partial length
200134 EIF2AK1 200134 Q9BQI3
Eukaryotic translation initiation factor 2-alpha kinase 1; EIF2AK1; HCR; HRI; KIAA1369
KINOMEscan Wild Type; Partial length
200072 CDC2L2 200072 Q9UQ88
Cyclin-dependent kinase 11A; CDC2L2; CDC2L3; CDK11A; CDK11-p110; CDK11-p46; CDK11-p58; MGC131975; p58GTA; PITSLRE
KINOMEscan Wild Type; Partial length
200071 CDC2L1 200071 P21127
Cyclin-dependent kinase 11B; CDC2L1; CDC2L2; CDK11; CDK11B; CDK11-p110; CDK11-p46; CDK11-p58; CLK-1; FLJ59152; p58; p58CDC2L1; p58CLK-1; PITSLRE; PK58
KINOMEscan Wild Type; Partial length
200040 ANKK1 200040 Q8NFD2
Ankyrin repeat and kinase domain containing 1; ANKK1; PKK2; SgK288
KINOMEscan Wild Type; Partial length
200070 CASK 200070 O14936
Calcium/calmodulin-dependent serine protein kinase (MAGUK family); CAGH39; CAMGUK; CASK; CMG; FGS4; FLJ22219; FLJ31914; LIN2; MICPCH; TNRC8
KINOMEscan Wild Type; Partial length
200069 CAMKK2 200069 Q96RR4
Calcium/calmodulin-dependent protein kinase kinase 2, beta; CAMKK; CAMKK2; CAMKKB; KIAA0787; MGC15254
KINOMEscan Wild Type; Partial length
200039 AMPK-alpha2 200039 P54646
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPK2; AMPKa2; AMPK-alpha2; PRKAA; PRKAA2
KINOMEscan Wild Type; Partial length
200237 M3K2 200237 Q9Y2U5
Mitogen-activated protein kinase kinase kinase 2; MAP3K2; MEKK2; MEKK2/MAP3K2; MEKK2B
KINOMEscan Wild Type; Partial length
200068 KKCC1 200068 Q8N5S9
Calcium/calmodulin-dependent protein kinase kinase 1, CaM-kinase IV kinase; CAMKK1; CAMKKA; DKFZp761M0423; MGC34095
KINOMEscan Wild Type; Partial length
200067 KCC4 200067 Q16566
Calcium/calmodulin-dependent protein kinase type IV; CAMK4; CaMK-GR; MGC36771
KINOMEscan Wild Type; Partial length
200066 CAMK2G 200066 Q13555
Calcium/calmodulin-dependent protein kinase II gamma; CAMK; CAMK2G; CAMKG; CAMK-II; FLJ16043; MGC26678
KINOMEscan Wild Type; Partial length
200122 EGFR 200122 P00533
Epidermal growth factor receptor (erythroblastic leukemia viral (v-erb-b) oncogene homolog, avian); EGFR; ERBB; ERBB1; HER1; mENA; PIG61
KINOMEscan Wild Type; Partial length
200065 KCC2D 200065 Q13557
Calcium/calmodulin-dependent protein kinase type II subunit delta; CaM kinase II subunit delta; CAMK2D; CAMKD; DKFZp686G23119; DKFZp686I2288; MGC44911
KINOMEscan Wild Type; Partial length
200038 AMPK-alpha1 200038 Q13131
Protein kinase, AMP-activated, alpha 2 catalytic subunit; AMPK; AMPKa1; AMPK-alpha1; MGC33776; MGC57364; PRKAA1
KINOMEscan Wild Type; Partial length
200037 ALK 200037 Q9UM73
Anaplastic lymphoma receptor tyrosine kinase; ALK; CD246; NBLST3; TFG/ALK
KINOMEscan Wild Type; Partial length
200119 DYRK1A 200119 Q13627
Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A; DYRK; DYRK1; DYRK1A; HP86; MNB; MNBH
KINOMEscan Wild Type; Partial length
200064 CAMK2B 200064 Q13554
Calcium/calmodulin-dependent protein kinase II beta; CAM2; CAMK2; CAMK2B; CAMKB; MGC29528
KINOMEscan Wild Type; Partial length
200117 DRAK1 200117 Q9UEE5
Serine/threonine kinase 17a; DRAK1; STK17A
KINOMEscan Wild Type; Partial length
200063 CAMK2A 200063 Q9UQM7
Calcium/calmodulin-dependent protein kinase II alpha; CAMK2A; CAMKA; KIAA0968
KINOMEscan Wild Type; Partial length
200036 AKT3 200036 Q9Y243
V-akt murine thymoma viral oncogene homolog 3 (protein kinase B, gamma); AKT3; Akt3/PKBg; DKFZp434N0250; PKBg; PKB-GAMMA; PRKBG; RAC-gamma; RAC-PK-gamma; STK-2
KINOMEscan Wild Type; Partial length
200116 DMPK2 200116 Q6DT37
CDC42 binding protein kinase gamma (DMPK-like); CDC42BPG; DMPK2; HSMDPKIN; KAPPA-200; MRCKgamma
KINOMEscan Wild Type; Partial length
200115 DMPK 200115 Q09013
Myotonin-protein kinase; Dystrophia myotonica-protein kinase; DM; DM1; DM1PK; DMK; MDPK; MT-PK
KINOMEscan Wild Type; Partial length
200062 CAMK1G 200062 Q96NX5
Calcium/calmodulin-dependent protein kinase IG; CAMK1G; CLICKIII; dJ272L16.1; VWS1
KINOMEscan Wild Type; Partial length