MLN-8054 KINOMEscan - Dataset (ID:20157)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200378 RIPK2 200378 O43353
Receptor-interacting serine/threonine-protein kinase 2; CARD3; CARDIAK; CCK; GIG30; RICK; RIP2; RIPK2
KINOMEscan Wild Type; Partial length
200379 RIPK4 200379 P57078
Receptor-interacting serine-threonine kinase 4; ANKK2; ANKRD3; DIK; MGC129992; MGC129993; PKK; RIP4
KINOMEscan Wild Type; Partial length
200381 ROCK1 200381 Q13464
Rho-associated protein kinase 1; Rho-associated, coiled-coil containing protein kinase 1; MGC131603; MGC43611; P160ROCK; PRO0435; ROCK1
KINOMEscan Wild Type; Partial length
200382 ROCK2 200382 O75116
Rho-associated protein kinase 2; Rho-associated, coiled-coil containing protein kinase 2; KIAA0619; ROCK2
KINOMEscan Wild Type; Partial length
200383 ROS1 200383 P08922
C-ros oncogene 1 , receptor tyrosine kinase; c-ros-1; MCF3; ROS; ROS1
KINOMEscan Wild Type; Partial length
200423 STK36 200423 Q9NRP7
Serine/threonine kinase 36, fused homolog (Drosophila); DKFZp434N0223; FU; Fused; KIAA1278; STK36
KINOMEscan Wild Type; Partial length
200390 RPS6KA4(Kin.Dom.1-N-terminal) 200390 O75676
Ribosomal protein S6 kinase, 90kDa, polypeptide 4; MSK2; RPS6KA4; RSK-B
KINOMEscan Kin.Dom.1-N-terminal Wild Type; Partial length
200392 RPS6KA4(Kin.Dom.2-C-terminal) 200392 O75676
Ribosomal protein S6 kinase, 90kDa, polypeptide 4; MSK2; MSK2~b; RPS6KA4; RSK-B
KINOMEscan Kin.Dom.2-C-terminal Wild Type; Partial length
200394 RPS6KA5(Kin.Dom.1-N-terminal) 200394 O75582
Ribosomal protein S6 kinase, 90kDa, polypeptide 5; MGC1911; MSK1; MSPK1; RLPK; RPS6KA5
KINOMEscan Kin.Dom.1-N-terminal Wild Type; Partial length
200396 RPS6KA5(Kin.Dom.2-C-terminal) 200396 O75582
Ribosomal protein S6 kinase, 90kDa, polypeptide 5; MGC1911; MSK1; MSK1~b; MSPK1; RLPK; RPS6KA5
KINOMEscan Kin.Dom.2-C-terminal Wild Type; Partial length
200399 RSK1(Kin.Dom.1-N-terminal) 200399 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KINOMEscan Kin.Dom.1-N-terminal) Wild Type; Partial length
200400 RSK1(Kin.Dom.2-C-terminal) 200400 Q15418
Ribosomal protein S6 kinase alpha 1; KS6A1
KINOMEscan Kin.Dom.2-C-terminal) Wild Type; Partial length
200401 RSK2(Kin.Dom.1-N-terminal) 200401 P51812
Ribosomal protein S6 kinase alpha 3; KS6A3; S6K-alpha-3; p90-RSK 3; MAPKAPK-1b; pp90RSK2
KINOMEscan Kin.Dom.1-N-terminal) Wild Type; Partial length
200444 TRKB 200444 Q16620
Neurotrophic tyrosine kinase, receptor, type 2; GP145-TrkB; NTRK2; TRKB
KINOMEscan Wild Type; Partial length
200402 RSK3(Kin.Dom.1-N-terminal) 200402 Q15349
Ribosomal protein S6 kinase, 90kDa, polypeptide 2; HU-2; MAPKAPK1C; p90RSK; p90-RSK3; pp90RSK3; RPS6KA2; RSK; RSK1; RSK1/p90RSK; RSK3; S6K-alpha; S6K-alpha2
KINOMEscan Kin.Dom.1-N-terminal) Wild Type; Partial length
200403 RSK3(Kin.Dom.2-C-terminal) 200403 Q15349
Ribosomal protein S6 kinase, 90kDa, polypeptide 2; HU-2; MAPKAPK1C; p90-RSK3; pp90RSK3; RPS6KA2; RSK; RSK1; RSK1~b; RSK3; S6K-alpha; S6K-alpha2
KINOMEscan Kin.Dom.2-C-terminal) Wild Type; Partial length
200404 RSK4(Kin.Dom.1-N-terminal) 200404 Q9UK32
Ribosomal protein S6 kinase alpha 6; S6K-alpha-6; p90-RSK 6; pp90RSK4
KINOMEscan Kin.Dom.1-N-terminal) Wild Type; Partial length
200405 RSK4(Kin.Dom.2-C-terminal) 200405 Q9UK32
Ribosomal protein S6 kinase alpha 6; S6K-alpha-6; p90-RSK 6; pp90RSK4
KINOMEscan Kin.Dom.2-C-terminal) Wild Type; Partial length
200406 S6K1 200406 P23443
Ribosomal protein S6 kinase, 70kDa, polypeptide 1; p70(S6K)-alpha; p70-alpha; p70S6K; p70-S6K; PS6K; RPS6KB1; S6K; S6K1; STK14A
KINOMEscan Wild Type; Partial length
200407 SBK1 200407 Q52WX2
SH3-binding domain kinase 1; Sbk; SBK1
KINOMEscan Wild Type; Partial length
200408 SgK110 200408 P0C264
Putative uncharacterized serine/threonine-protein kinase (Sugen kinase 110); SgK110
KINOMEscan Wild Type; Partial length
200409 SGK3 200409 Q96BR1
Serine/threonine-protein kinase Sgk3; Serum/glucocorticoid-regulated kinase 3; CISK; DKFZp781N0293; SGKL
KINOMEscan Wild Type; Partial length
200410 SIK1 200410 P57059
Serine/threonine-protein kinase SIK1; salt-inducible kinase 1; MSK; SIK; SIK1; SNF1LK
KINOMEscan Wild Type; Partial length
200412 SLK 200412 Q9H2G2
STE20-like serine/threonine-protein kinase; CTCL tumor antigen se20-9; bA16H23.1; KIAA0204; LOSK; MGC133067; se20-9; SLK; STK2
KINOMEscan Wild Type; Partial length
200413 SNARK 200413 Q9H093
NUAK family, SNF1-like kinase, 2; DKFZp434J037; DKFZp686F01113; FLJ90349; NUAK2; SNARK
KINOMEscan Wild Type; Partial length