MLN-8054 KINOMEscan - Dataset (ID:20157)
Proteins Studied
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LINCS ID | Name | HMS LINCS ID | UniProt ID | Alternative Names | Provider | Mutation | Phosphlorylation State | Domain | Protein Description |
---|---|---|---|---|---|---|---|---|---|
200241 | M4K3 | 200241 | Q8IVH8 | Mitogen-activated protein kinase kinase kinase kinase 3; GLK; KHS2; MAP4K3; MAPKKKK3; MEKKK3; RAB8IPL1 | KINOMEscan | Wild Type; Partial length | |||
200186 | HIPK1 | 200186 | Q86Z02 | Homeodomain interacting protein kinase 1; HIPK1; KIAA0630; MGC26642; MGC33446; MGC33548; Myak; Nbak2 | KINOMEscan | Wild Type; Partial length | |||
200187 | HIPK2 | 200187 | Q9H2X6 | Homeodomain interacting protein kinase 2; DKFZp686K02111; FLJ23711; HIPK2; PRO0593 | KINOMEscan | Wild Type; Partial length | |||
200188 | HIPK3 | 200188 | Q9H422 | Homeodomain interacting protein kinase 3; DYRK6; FIST3; HIPK3; PKY; YAK1 | KINOMEscan | Wild Type; Partial length | |||
200189 | HIPK4 | 200189 | Q8NE63 | Homeodomain interacting protein kinase 4; FLJ32818; HIPK4 | KINOMEscan | Wild Type; Partial length | |||
200100 | KC1G1 | 200100 | Q9HCP0 | Casein kinase I isoform gamma-1; CK1g1; CSNK1G1 | KINOMEscan | Wild Type; Partial length | |||
200191 | HUNK | 200191 | P57058 | Hormonally up-regulated Neu-associated kinase; HUNK | KINOMEscan | Wild Type; Partial length | |||
200192 | ICK | 200192 | Q9UPZ9 | Intestinal cell (MAK-like) kinase; ECO; ICK; KIAA0936; LCK2; MGC46090; MRK | KINOMEscan | Wild Type; Partial length | |||
200193 | IGF1R | 200193 | P08069 | Insulin-like growth factor 1 receptor; CD221; IGF1R; IGFIR; IGFR; JTK13; MGC142170; MGC142172; MGC18216 | KINOMEscan | Wild Type; Partial length | |||
200287 | NEK11 | 200287 | Q8NG66 | NIMA (never in mitosis gene a)-related kinase 11; FLJ23495; NEK11 | KINOMEscan | Wild Type; Partial length | |||
200288 | NEK2 | 200288 | P51955 | Serine/threonine-protein kinase Nek2; NIMA (never in mitosis gene a)-related kinase 2; HsPK21; NEK2; NEK2A; NLK1 | KINOMEscan | Wild Type; Partial length | |||
200056 | PTK6 | 200056 | Q13882 | Protein tyrosine kinase 6; BRK; FLJ42088; PTK6 | KINOMEscan | Wild Type; Partial length | |||
200197 | INSR | 200197 | P06213 | Insulin receptor; CD220; HHF5; INSR; IR | KINOMEscan | Wild Type; Partial length | |||
200198 | INSRR | 200198 | P14616 | Insulin receptor-related receptor; INSRR; IRR | KINOMEscan | Wild Type; Partial length | |||
200199 | IRAK1 | 200199 | P51617 | Interleukin-1 receptor-associated kinase 1 | KINOMEscan | Wild Type; Partial length | |||
200200 | IRAK3 | 200200 | Q9Y616 | Interleukin-1 receptor-associated kinase 3; ASRT5; FLJ13601; IRAK3; IRAKM | KINOMEscan | Wild Type; Partial length | |||
200201 | IRAK4 | 200201 | Q9NWZ3 | Interleukin-1 receptor-associated kinase 4; IPD1; NY-REN-64; REN64 | KINOMEscan | Wild Type; Partial length | |||
200202 | ITK | 200202 | Q08881 | IL2-inducible T-cell kinase; EMT; ITK; LYK; MGC126257; MGC126258; PSCTK2 | KINOMEscan | Wild Type; Partial length | |||
200203 | JAK1(JH1domain-catalytic) | 200203 | P23458 | Janus kinase 1; JAK1; JAK1A; JAK1B; JAK1-catalytic; JTK3 | KINOMEscan | JH1domain-catalytic | Wild Type; Partial length | ||
200204 | JAK1(JH2domain-pseudokinase) | 200204 | P23458 | Janus kinase 1; JAK1; JAK1~b; JAK1A; JAK1B; JAK1-pseudokinase; JTK3 | KINOMEscan | JH2domain-pseudokinase | Wild Type; Partial length | ||
200207 | JAK2(JH1domain-catalytic) | 200207 | O60674 | Janus kinase 2; JAK2; JAK2-catalytic; JTK10 | KINOMEscan | JH1domain-catalytic | Wild Type; Partial length | ||
200209 | JAK3(JH1domain-catalytic) | 200209 | P52333 | Tyrosine-protein kinase JAK3; Janus kinase 3; JAK-3; L-JAK | KINOMEscan | JH1domain-catalytic | Wild Type; Partial length | ||
200108 | DAPK3 | 200108 | O43293 | Death-associated protein kinase 3; DAPK3; FLJ36473; ZIP; ZIPK | KINOMEscan | Wild Type; Partial length | |||
200109 | DCLK1 | 200109 | O15075 | Serine/threonine-protein kinase DCLK1; CL1; CLICK1; DCAMKL1; DCDC3A; DCLK; DCLK1; KIAA0369 | KINOMEscan | Wild Type; Partial length | |||
200346 | PKMYT1 | 200346 | Q99640 | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase; Protein kinase, membrane associated tyrosine/threonine 1; DKFZp547K1610; FLJ20093; MYT1 | KINOMEscan | Wild Type; Partial length |